SCHEMBL8971437

SCHEMBL8971437

COc1ccc(COc2cc(N)c(Cl)cc2CC(=O)CCCN2CCCCC2)cc1OC

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 11/20 0.56
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
CYP3A4 P08684 2/20 0.50
ALDH1A1 P00352 2/20 0.50
CYP2D6 P10635 2/20 0.50
HTR3A P46098 1/20 0.50
GLA P06280 1/20 0.47
CYP2C9 P11712 1/20 0.41
TSHR P16473 1/20 0.41
ACHE P22303 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8971588 0.90 HTR4 (0.54) HTR4MEN1KMT2ACYP3A4ALDH1A1
SCHEMBL8971888 0.88 HTR4 (0.56) HTR4MEN1KMT2ACYP3A4ALDH1A1
SCHEMBL8971037 0.88 HTR4 (0.56) HTR4MEN1KMT2ACYP3A4ALDH1A1
SCHEMBL8971367 0.87 HTR4 (0.69) HTR4MEN1KMT2ACYP3A4ALDH1A1
SCHEMBL8971616 0.86 HTR4 (0.54) HTR4MEN1KMT2ACYP3A4ALDH1A1
Hydrochloric Acid SCHEMBL3684761 0.86 HTR4 (0.68) HTR4MEN1KMT2ACYP3A4ALDH1A1
Hydrochloric Acid SCHEMBL8971612 0.85 HTR4 (0.66) HTR4MEN1KMT2ACYP3A4ALDH1A1
Hydrochloric Acid SCHEMBL8971911 0.85 HTR4 (0.52) HTR4MEN1KMT2ACYP3A4ALDH1A1
SCHEMBL7350017 0.83 HTR4 (0.75) HTR4MEN1KMT2ACYP3A4ALDH1A1
Hydrochloric Acid SCHEMBL8971067 0.82 HTR4 (0.57) HTR4MEN1KMT2ACYP3A4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0700383-A1 NOVEL 1-PHENYLALKANONE 5-HT 4? RECEPTOR LIGANDS SYNTEX (U.S.A.) INC. (US) 1996-03-13 EP disclosed