SCHEMBL8973563

SCHEMBL8973563

O=C1c2ccccc2S(=O)(=O)N1CCCBr

nearest known ligand 0.72

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 10/20 0.72
CA12 O43570 10/20 0.72
CA2 P00918 3/20 0.67
ELANE P08246 1/20 0.61
HDAC1 Q13547 1/20 0.59
HDAC2 Q92769 1/20 0.59
HPGD P15428 1/20 0.58
DRD2 P14416 3/20 0.58
DRD4 P21917 1/20 0.58
DRD5 P21918 1/20 0.58
DRD3 P35462 1/20 0.58
ACHE P22303 1/20 0.58
ALDH1A1 P00352 1/20 0.57
CYP2C19 P33261 1/20 0.57
HTR1A P08908 2/20 0.56
HTR2A P28223 2/20 0.56
HTR7 P34969 2/20 0.56
HTR6 P50406 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6324557 0.95 CA9 (0.73) CA9CA12CA2ELANEHDAC1
SCHEMBL4033933 0.94 CA9 (0.71) CA9CA12CA2ELANEHDAC1
SCHEMBL5354797 0.94 CA9 (0.71) CA9CA12CA2ELANEHDAC1
SCHEMBL9437884 0.90 CA12 (0.71) CA9CA12CA2ELANEHPGD
SCHEMBL30872949 0.90 CA12 (0.71) CA9CA12CA2ELANEHPGD
SCHEMBL7932914 0.85 CA9 (0.74) CA9CA12CA2ELANEHDAC1
SCHEMBL7903703 0.84 CA9 (1.00) CA9CA12CA2ELANEHDAC1
SCHEMBL17372964 0.84 CA9 (0.72) CA9CA12CA2ELANEHDAC1
SCHEMBL5120710 0.84 CA9 (0.72) CA9CA12CA2ELANEHDAC1
SCHEMBL7281348 0.83 CA12 (0.69) CA9CA12CA2ELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5585392-A TREATING OR PREVENTING STROKES BAYER AKTIENGESELLSCHAFT (DE) 1996-12-17 US disclosed
US-5506246-A Method for treating depression using substituted aminomethyltetralins and their heterocyclic analogues BAYER AKTIENGESELLSCHAFT (DE) 1996-04-09 US disclosed
US-5463105-A Therapy for cardiovascular, nervous system disorders BAYER AKTIENGESELLSCHAFT (DE) 1995-10-31 US disclosed
US-5453437-A 1,3-disubstituted pyrrolidines BAYER AKTIENGESELLSCHAFT (DE) 1995-09-26 US disclosed
US-5300523-A Binding serotonin receptors, treating nervous system disorders BAYER AKTIENGESELLSCHAFT (DE) 1994-04-05 US disclosed
US-5298513-A Serotonin antagonist BAYER AKTIENGESELLSCHAFT (DE) 1994-03-29 US disclosed
US-5296477-A Antidepressants ADIR ET COMPAGNIE (FR) 1994-03-22 US disclosed
US-5274097-A A 1-N-heterocyclic alkylene-3-carbo or heterocyclic ring oxypyrrolidine derivative BAYER AKTIENGESELLSCHAFT (DE) 1993-12-28 US disclosed
US-5268381-A Antidepressant or anxiolytic compound ADIR ET COMPAGNIE (FR) 1993-12-07 US disclosed
US-5196434-A Antidepressants, anxiolytic agents ADIR ET COMPAGNIE (FR) 1993-03-23 US disclosed
US-5153225-A For treating disorders of the central nervous system, cardiovascular system and intestinal tract BAYER AKTIENGESELLSCHAFT (DE) 1992-10-06 US disclosed
US-5137901-A For binding 5-HT 1 receptors; treating central nervous system disorders BAYER AKTIENGESELLSCHAFT (DE) 1992-08-11 US disclosed
EP-0478446-A1 Heterocyclic alkylamines, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1992-04-01 EP disclosed
US-5021438-A Having affinity for 5-hydroxytryptamine receptors; treating central nervous system and cardiovascular disorders BAYER AKTIENGESELLSCHAFT (DE) 1991-06-04 US disclosed
US-4880802-A CENTRAL NERVOUS SYSTEM BAYER AKTIENGESELLSCHAFT (DE) 1989-11-14 US disclosed