SCHEMBL8974180

SCHEMBL8974180

CC1(C)C=C(c2ccc(S(C)(=O)=O)cc2)C(c2ccc(F)nc2)=C1

nearest known ligand 0.50

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 17/20 0.50
PTGS1 P23219 6/20 0.50
MMP2 P08253 1/20 0.41
MMP9 P14780 1/20 0.41
MMP13 P45452 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974088 0.89 PTGS2 (0.50) PTGS2PTGS1MMP2MMP9MMP13
SCHEMBL8974247 0.87 PTGS2 (0.45) PTGS2PTGS1MMP2MMP9MMP13
SCHEMBL9118925 0.86 PTGS2 (0.70) PTGS2PTGS1MMP2MMP9MMP13
SCHEMBL8974363 0.85 PTGS2 (0.47) PTGS2PTGS1MMP2MMP9MMP13
SCHEMBL8974501 0.85 PTGS2 (0.47) PTGS2PTGS1MMP2MMP9MMP13
SCHEMBL8973837 0.85 PTGS2 (0.47) PTGS2PTGS1MMP2MMP9MMP13
SCHEMBL8974336 0.84 KCNH2 (0.54) PTGS2PTGS1
SCHEMBL8974812 0.84 PTGS2 (0.49) PTGS2PTGS1MMP2MMP9MMP13
SCHEMBL9126561 0.84 PTGS2 (0.63) PTGS2PTGS1MMP2MMP9MMP13
SCHEMBL9118108 0.84 PTGS2 (0.63) PTGS2PTGS1MMP2MMP9MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO claimed
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed