SCHEMBL8974285

SCHEMBL8974285

Cc1ccc(C2=CC(C)(C(F)(F)F)C=C2c2ccc(S(C)(=O)=O)cc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 17/20 0.49
PTGS1 P23219 5/20 0.49
CYP2C9 P11712 1/20 0.44
KIF11 P52732 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974303 0.88 PTGS2 (0.64) PTGS2PTGS1
SCHEMBL8974500 0.87 PTGS2 (0.52) PTGS2PTGS1
SCHEMBL8974455 0.87 PTGS2 (0.55) PTGS2PTGS1KIF11
SCHEMBL9116379 0.76 PTGS2 (0.74) PTGS2PTGS1
SCHEMBL12341698 0.74 PTGS2 (0.68) PTGS2PTGS1
SCHEMBL8973922 0.74 PTGS2 (0.66) PTGS2PTGS1
SCHEMBL8974161 0.74 PTGS2 (0.57) PTGS2PTGS1KIF11
SCHEMBL8975150 0.73 PTGS2 (0.51) PTGS2PTGS1
SCHEMBL8974655 0.73 PTGS2 (0.56) PTGS2PTGS1KIF11
SCHEMBL12807 0.72 GAA (0.65) PTGS2PTGS1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed