SCHEMBL8974642

SCHEMBL8974642

CC(CO)N1CCOC(COc2cccc(Cl)c2)C1

nearest known ligand 0.59

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 4/20 0.59
DRD4 P21917 8/20 0.52
ACLY P53396 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8857239 0.86 HRH3 (0.55) HRH3DRD4ACLY
SCHEMBL14018436 0.81 DRD4 (0.57) HRH3DRD4
SCHEMBL8857234 0.78 DRD4 (0.57) DRD4
SCHEMBL8975092 0.77 PPARG (0.47) HRH3DRD4
SCHEMBL8974671 0.77 GRM2 (0.60)
SCHEMBL8974668 0.77 GRM2 (0.60)
SCHEMBL8975043 0.77 GRM2 (0.60)
SCHEMBL8975210 0.77 GRM2 (0.60)
SCHEMBL8974912 0.77 GRM2 (0.60)
SCHEMBL8975062 0.77 GRM2 (0.60)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1065532-C Thiazolidine and oxazolidine derivatives, their preparation and their medical use SANKYO CO (JP) 2001-05-09 CN disclosed
US-5578620-A TREATMENT OF DIABETES AND HYPERLIPEMIA SANKYO COMPANY, LIMITED (JP) 1996-11-26 US disclosed
CN-1132750-A Thiazolidine and oxazolidine derivatives, their preparation and their medical use SANKYO CO (JP) 1996-10-09 CN disclosed
EP-0678511-A2 Thiazolidine and oxazolidine derivatives, their preparation and their medical use SANKYO COMPANY LIMITED (JP) 1995-10-25 EP disclosed