SCHEMBL8975717

SCHEMBL8975717

C#CCCCCOCC#C

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.50
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
MAPT P10636 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
HSD17B10 Q99714 1/20 0.34
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31
CA2 P00918 1/20 0.30
CA9 Q16790 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17186655 0.89 TSHR (0.58) TSHRHSD17B10
SCHEMBL11569672 0.86 TSHR (0.56) TSHRHSD17B10
SCHEMBL11572476 0.86 TSHR (0.56) TSHRHSD17B10
SCHEMBL26205671 0.86 TSHR (0.56) TSHRHSD17B10
SCHEMBL11571608 0.86 TSHR (0.56) TSHRHSD17B10
SCHEMBL9585705 0.86 CYP1A2 (0.39) TSHRCYP1A2CYP2D6MAPTCYP2C9
SCHEMBL766061 0.86 TSHR (0.56) TSHRHSD17B10
SCHEMBL11572511 0.86 TSHR (0.56) TSHRHSD17B10
SCHEMBL26205674 0.86 TSHR (0.56) TSHRHSD17B10
SCHEMBL26205673 0.86 TSHR (0.56) TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0543919-B1 USE OF HETEROCYCLIC AMINO-ALCOHOL COMPOUNDS IN THE MANUFACTURE OF A MEDICAMENT FOR TREATMENT OF CNS DISEASES SEARLE & CO (US) 1996-04-10 EP claimed