SCHEMBL8976231

SCHEMBL8976231

O=[N+]([O-])c1ccc2ncnc(Nc3ccc4ncccc4c3)c2c1

nearest known ligand 0.69

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EGFR P00533 10/20 0.69
ALK Q9UM73 1/20 0.66
ALDH1A1 P00352 3/20 0.62
MAPT P10636 3/20 0.62
HTT P42858 3/20 0.62
MEN1 O00255 1/20 0.62
KMT2A Q03164 1/20 0.62
L3MBTL1 Q9Y468 1/20 0.60
ABCG2 Q9UNQ0 3/20 0.58
EIF2AK2 P19525 1/20 0.56
ERBB2 P04626 1/20 0.55
ERBB4 Q15303 1/20 0.55
GAA P10253 1/20 0.51
NCOA1 Q15788 1/20 0.51
NCOA3 Q9Y6Q9 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30638097 0.83 EGFR (0.59) EGFRALKMAPTHTTABCG2
SCHEMBL157043 0.83 EGFR (0.59) EGFRALKMAPTHTTABCG2
SCHEMBL1192454 0.82 EGFR (1.00) EGFRALKALDH1A1MAPTHTT
SCHEMBL8976408 0.81 EGFR (1.00) EGFRALDH1A1MAPTHTTERBB2
SCHEMBL4587672 0.81 ALK (0.79) EGFRALKALDH1A1MAPTHTT
SCHEMBL159107 0.80 EGFR (0.68) EGFRABCG2ERBB2ERBB4
SCHEMBL18349251 0.80 EGFR (0.77) EGFRALKALDH1A1MAPTHTT
SCHEMBL3244626 0.80 ALK (0.77) EGFRALKALDH1A1MAPTHTT
Hydrochloric Acid SCHEMBL8976403 0.79 EGFR (0.67) EGFRALKALDH1A1MAPTHTT
SCHEMBL8976740 0.79 EGFR (0.69) EGFRALKALDH1A1MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5580870-A ANTICARCINOGENIC AGENTS ZENECA LIMITED (GB) 1996-12-03 US disclosed
EP-0602851-B1 Quinazoline derivatives ZENECA LTD (GB) 1996-10-09 EP disclosed
CN-1094043-A Quinazoline derivant ZENECA LTD (GB) 1994-10-26 CN disclosed
EP-0602851-A1 Quinazoline derivatives ZENECA LIMITED (GB) 1994-06-22 EP disclosed