SCHEMBL8976740

SCHEMBL8976740

O=[N+]([O-])c1ccc2ncnc(Nc3ccc4[nH]ncc4c3)c2c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 7/20 0.69
ALK Q9UM73 1/20 0.62
MKNK1 Q9BUB5 2/20 0.61
RET P07949 1/20 0.60
MAPT P10636 3/20 0.59
ALDH1A1 P00352 2/20 0.59
HTT P42858 2/20 0.59
MEN1 O00255 1/20 0.59
KMT2A Q03164 1/20 0.59
L3MBTL1 Q9Y468 1/20 0.57
POLB P06746 1/20 0.56
MAOB P27338 1/20 0.56
NOS1 P29475 1/20 0.56
RAF1 P04049 1/20 0.55
BRAF P15056 1/20 0.55
EIF2AK2 P19525 1/20 0.53
ABCG2 Q9UNQ0 1/20 0.52
HSF1 Q00613 1/20 0.52
ROCK2 O75116 1/20 0.50
ROCK1 Q13464 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8976301 0.99 EGFR (0.68) EGFRALKMKNK1RETMAPT
Hydrochloric Acid SCHEMBL8976403 0.83 EGFR (0.67) EGFRALKMAPTALDH1A1HTT
SCHEMBL173234 0.82 EGFR (0.60) EGFRMKNK1RETRAF1BRAF
SCHEMBL8096187 0.82 EGFR (1.00) EGFRMKNK1RETRAF1BRAF
SCHEMBL3585835 0.82 ABCG2 (0.70) ABCG2ROCK2
SCHEMBL3587306 0.81 ABCG2 (0.62) MAPTPOLBMAOBNOS1ABCG2
SCHEMBL15050482 0.80 RET (0.76) EGFRMKNK1RETL3MBTL1RAF1
SCHEMBL2835747 0.79 EGFR (0.74) EGFRMKNK1RETRAF1BRAF
SCHEMBL29516907 0.79 EGFR (0.74) EGFRMKNK1RETRAF1BRAF
SCHEMBL8976231 0.79 EGFR (0.69) EGFRALKMAPTALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5580870-A ANTICARCINOGENIC AGENTS ZENECA LIMITED (GB) 1996-12-03 US disclosed
EP-0602851-B1 Quinazoline derivatives ZENECA LTD (GB) 1996-10-09 EP disclosed
EP-0602851-A1 Quinazoline derivatives ZENECA LIMITED (GB) 1994-06-22 EP disclosed