SCHEMBL8978402

SCHEMBL8978402

CCCn1c2ncnc-2cnc1C1CC1.CCn1cnc(NC2CCCC2)c2nc(C(C)C)nc1-2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 7/20 0.37
ADORA3 P0DMS8 6/20 0.37
ADORA2A P29274 6/20 0.37
ADORA2B P29275 6/20 0.37
CTSL P07711 1/20 0.34
CTSB P07858 1/20 0.34
FLT3 P36888 4/20 0.33
PLK4 O00444 1/20 0.33
CHEK1 O14757 1/20 0.33
MAPK13 O15264 1/20 0.33
DAPK3 O43293 1/20 0.33
PRKCG P05129 1/20 0.33
CDK1 P06493 1/20 0.33
LYN P07948 1/20 0.33
PIM1 P11309 1/20 0.33
PRKACA P17612 1/20 0.33
CDK2 P24941 1/20 0.33
MARK3 P27448 1/20 0.33
MAPK1 P28482 1/20 0.33
AKT2 P31751 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1388167 0.81 CHRM3 (0.40) ADORA1ADORA3ADORA2AADORA2BCTSL
Hydrochloric Acid SCHEMBL7029936 0.80 CHRM3 (0.39) ADORA1ADORA3ADORA2AADORA2BCTSL
SCHEMBL1387953 0.79 CTSL (0.47) ADORA1ADORA3ADORA2AADORA2BCTSL
Hydrochloric Acid SCHEMBL7028301 0.79 CTSL (0.46) ADORA1ADORA3ADORA2AADORA2BCTSL
SCHEMBL1388124 0.79 CTSL (0.48) ADORA1ADORA3ADORA2AADORA2BCTSL
SCHEMBL8396714 0.78 CTSL (0.37) ADORA1ADORA3ADORA2AADORA2BCTSL
Hydrochloric Acid SCHEMBL7023573 0.78 CTSL (0.47) ADORA1ADORA3ADORA2AADORA2BCTSL
SCHEMBL1387905 0.70 CHRM3 (0.48) ADORA1ADORA3ADORA2AADORA2BCTSL
Hydrochloric Acid SCHEMBL7027686 0.69 CHRM3 (0.47) ADORA1ADORA3ADORA2AADORA2BCTSL
SCHEMBL8397096 0.69 CTSL (0.41) ADORA1ADORA3ADORA2AADORA2BCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705265-A1 NOVEL CHEMICAL COMPOUNDS HAVING PDE-IV INHIBITION ACTIVITY Euroceltique S.A. (LU) 1996-04-10 EP claimed