SCHEMBL8978653

SCHEMBL8978653

CCn1c(-c2cc(OC)ccc2N)n[nH]c1=S

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.58
ALDH1A1 P00352 7/20 0.58
HPGD P15428 4/20 0.58
GAA P10253 3/20 0.53
TDP1 Q9NUW8 3/20 0.53
KMT2A Q03164 2/20 0.53
HSD17B10 Q99714 2/20 0.53
MAPT P10636 2/20 0.53
GLA P06280 1/20 0.53
HTT P42858 1/20 0.51
GFER P55789 3/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
PKM P14618 1/20 0.50
MTNR1B P49286 1/20 0.47
MAPK1 P28482 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8978588 0.82 ALDH1A1 (0.62) KDM4EALDH1A1HPGDGAATDP1
SCHEMBL8978548 0.82 APOBEC3G (0.62) KDM4EALDH1A1HPGDGAATDP1
SCHEMBL8978524 0.80 ALDH1A1 (0.50) KDM4EALDH1A1HPGDGAAKMT2A
SCHEMBL8978559 0.79 GFER (0.74) KDM4EALDH1A1HPGDGAATDP1
SCHEMBL8978608 0.79 ALDH1A1 (0.74) KDM4EALDH1A1HPGDGAATDP1
SCHEMBL8978556 0.78 ALDH1A1 (0.69) KDM4EALDH1A1HPGDGAATDP1
SCHEMBL8978579 0.76 KDM4E (0.54) KDM4EALDH1A1HPGDGAATDP1
SCHEMBL8978540 0.74 ALDH1A1 (0.59) KDM4EALDH1A1HPGDGAATDP1
SCHEMBL1544591 0.74 KDM4E (0.52) KDM4EALDH1A1HPGDGAATDP1
SCHEMBL8978530 0.73 GFER (0.74) KDM4EALDH1A1HPGDGAATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5489598-A INHIBITS ADHESION OF MAC-1 TO ENDOTHELIAL CELLS, USEFUL FOR TREATING GASTRITIS INDUCED BY NONSTEROIDANTIINFLAMMATORY DRUGS IMFLAMMATORY BOWEL DISEASE OF ULCERATIVE COLITIS WARNER-LAMBERT COMPANY (US) 1996-02-06 US disclosed