SCHEMBL8980359

SCHEMBL8980359

O=C(Nc1ccc2nc(-c3ccccc3)ccc2c1)c1ccccc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.69
RAB9A P51151 5/20 0.69
PLAU P00749 2/20 0.69
PABPC1 P11940 1/20 0.63
KMT2A Q03164 4/20 0.61
MEN1 O00255 3/20 0.61
SMN1; SMN2 Q16637 2/20 0.61
TP53 P04637 1/20 0.61
MAPT P10636 1/20 0.61
TRPV1 Q8NER1 1/20 0.55
ADORA1 P30542 2/20 0.55
PTPN1 P18031 2/20 0.55
KDR P35968 1/20 0.55
PTPN2 P17706 1/20 0.55
ADORA3 P0DMS8 1/20 0.52
F2 P00734 1/20 0.52
PLG P00747 1/20 0.52
KLKB1 P03952 1/20 0.52
PRSS1 P07477 1/20 0.52
HTT P42858 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26613421 0.87 NPC1 (0.55) NPC1RAB9APLAUPABPC1KMT2A
SCHEMBL26613556 0.84 PLAU (0.52) NPC1RAB9APLAUPABPC1MAPT
SCHEMBL26613551 0.84 KMT2A (0.59) NPC1RAB9APABPC1KMT2AMEN1
SCHEMBL2176831 0.82 NPC1 (1.00) NPC1RAB9APLAUPABPC1KMT2A
SCHEMBL26613478 0.81 ADORA1 (0.57) NPC1RAB9APLAUKMT2AMEN1
SCHEMBL20741553 0.80 NPC1 (0.51) NPC1RAB9APLAUPABPC1KMT2A
SCHEMBL29746102 0.79 NPC1 (0.53) NPC1RAB9APLAUKMT2AMEN1
SCHEMBL26613566 0.79 NPC1 (0.53) NPC1RAB9APLAUKMT2AMEN1
SCHEMBL3202307 0.79 NPC1 (0.46) NPC1RAB9APLAUPABPC1KMT2A
SCHEMBL24609656 0.79 SERPINE1 (0.53) NPC1RAB9APLAUKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5571822-A AMINO-2-PHENYL-4-QUINOLONE DERIVATIVES THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1996-11-05 US disclosed
WO-1996010563-A1 2-ARYL-4-QUINOLONES AS ANTITUMOR COMPOUNDS THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1996-04-11 WO disclosed