SCHEMBL8980648

SCHEMBL8980648

CC(=O)c1cccc(C(=O)OCc2ccccc2)c1OCc1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.58
TDP1 Q9NUW8 4/20 0.56
L3MBTL1 Q9Y468 4/20 0.54
TSHR P16473 2/20 0.54
CYP3A4 P08684 1/20 0.54
MAPK1 P28482 1/20 0.54
POLB P06746 1/20 0.52
CASP3 P42574 1/20 0.52
RAB9A P51151 1/20 0.52
SENP8 Q96LD8 1/20 0.52
SENP7 Q9BQF6 1/20 0.52
SENP6 Q9GZR1 1/20 0.52
MAOB P27338 3/20 0.50
SLC6A2 P23975 1/20 0.50
SLC6A3 Q01959 1/20 0.50
KMT2A Q03164 1/20 0.50
HTT P42858 2/20 0.48
MAPT P10636 2/20 0.48
CYP2C9 P11712 2/20 0.48
CYP2C19 P33261 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15716659 0.92 ALDH1A1 (0.67) ALDH1A1TDP1L3MBTL1TSHRCYP3A4
SCHEMBL8980650 0.86 MAOB (0.54) ALDH1A1TDP1L3MBTL1MAPK1MAOB
SCHEMBL16789584 0.84 ALDH1A1 (0.64) ALDH1A1TDP1L3MBTL1TSHRCYP3A4
SCHEMBL2640064 0.84 ALDH1A1 (0.74) ALDH1A1TDP1L3MBTL1TSHRCYP3A4
SCHEMBL31354660 0.84 ALDH1A1 (0.64) ALDH1A1TDP1L3MBTL1TSHRCYP3A4
SCHEMBL21022925 0.84 ALDH1A1 (0.59) ALDH1A1TDP1L3MBTL1TSHRCYP3A4
SCHEMBL1317303 0.82 POLB (0.59) ALDH1A1TDP1L3MBTL1TSHRCYP3A4
SCHEMBL4145578 0.82 ALDH1A1 (0.58) ALDH1A1TDP1L3MBTL1TSHRCYP3A4
SCHEMBL4240186 0.82 TDP1 (0.64) ALDH1A1TDP1L3MBTL1TSHRCYP3A4
SCHEMBL8489879 0.82 MAPT (0.57) TDP1L3MBTL1MAPK1MAOBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1132508-A Piperazine derivatives REORDATI IND CHIMICA E FARMACE (CH) 1996-10-02 CN disclosed
EP-0711288-A1 PIPERAZINE DERIVATIVES AS ALPHA 1A-ADRENERGIC RECEPTOR ANTAGONISTS RECORDATI INDUSTRIA CHIMICA E FARMACEUTICA S.p.a. (IT) 1996-05-15 EP disclosed
WO-1995004049-A1 PIPERAZINE DERIVATIVES AS α1A-ADRENERGIC RECEPTOR ANTAGONISTS RECORDATI S.A., CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1995-02-09 WO disclosed