SCHEMBL8980684

SCHEMBL8980684

CS(=O)(=O)OC(=O)c1ccccc1OCc1ccccc1Cl

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.54
MEN1 O00255 1/20 0.54
POLB P06746 1/20 0.54
KMT2A Q03164 1/20 0.54
HTT P42858 2/20 0.53
TP53 P04637 1/20 0.53
SGMS2 Q8NHU3 1/20 0.49
FABP4 P15090 3/20 0.49
FABP5 Q01469 3/20 0.49
LMNA P02545 2/20 0.48
L3MBTL1 Q9Y468 2/20 0.48
TDP1 Q9NUW8 1/20 0.48
KDM4E B2RXH2 1/20 0.48
MCL1 Q07820 1/20 0.48
CASP3 P42574 2/20 0.46
SENP8 Q96LD8 2/20 0.46
SENP7 Q9BQF6 2/20 0.46
SENP6 Q9GZR1 2/20 0.46
TRPM8 Q7Z2W7 2/20 0.46
MAOA P21397 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8980620 0.85 PLA2G1B (0.46) ALDH1A1MEN1POLBKMT2AHTT
SCHEMBL8980678 0.83 TP53 (0.66) ALDH1A1MEN1POLBKMT2AHTT
SCHEMBL8980628 0.81 ABCB1 (0.50) ALDH1A1MEN1KMT2A
SCHEMBL8278415 0.80 TP53 (0.61) ALDH1A1MEN1POLBKMT2AHTT
SCHEMBL1388155 0.79 HTT (0.77) ALDH1A1MEN1POLBKMT2AHTT
SCHEMBL8980720 0.79 ENPP2 (0.54) ALDH1A1SGMS2KDM4ETRPM8MAOA
SCHEMBL13690028 0.75 TP53 (0.54) ALDH1A1MEN1POLBKMT2AHTT
Water SCHEMBL8980731 0.74 KDM4E (0.47) POLBHTTL3MBTL1KDM4E
SCHEMBL27738026 0.74 TSHR (0.44) ALDH1A1KMT2AHTTTP53LMNA
Water SCHEMBL8980780 0.73 CAPN1 (0.49) HTTLMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0711288-A1 PIPERAZINE DERIVATIVES AS ALPHA 1A-ADRENERGIC RECEPTOR ANTAGONISTS RECORDATI INDUSTRIA CHIMICA E FARMACEUTICA S.p.a. (IT) 1996-05-15 EP disclosed
WO-1995004049-A1 PIPERAZINE DERIVATIVES AS α1A-ADRENERGIC RECEPTOR ANTAGONISTS RECORDATI S.A., CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1995-02-09 WO disclosed