SCHEMBL8985233

SCHEMBL8985233

O=C(O)C1CCc2nccn2C1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 8/20 0.53
NAMPT P43490 2/20 0.41
ADRA1D P25100 3/20 0.41
ADRA1B P35368 1/20 0.40
KDM4E B2RXH2 1/20 0.39
CYP2C19 P33261 1/20 0.39
NOTUM Q6P988 5/20 0.37
NEK2 P51955 1/20 0.36
ADRA2A P08913 1/20 0.35
CDK9 P50750 1/20 0.35
GABRP O00591 1/20 0.35
GABRD O14764 1/20 0.35
GABRA1 P14867 1/20 0.35
GABRB1 P18505 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRR1 P24046 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
GABRA3 P34903 1/20 0.35
GABRA2 P47869 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL31132960 0.98 ADRA1A (0.51) ADRA1ANAMPTADRA1DADRA1BKDM4E
SCHEMBL16112524 0.85 ADRA1A (0.48) ADRA1ANAMPTADRA1DADRA1BKDM4E
SCHEMBL30630523 0.79 ADRA1A (0.52) ADRA1ANAMPTADRA1DADRA1BADRA2A
SCHEMBL16067955 0.78 POLB (0.46) ADRA1AKDM4ECYP2C19
SCHEMBL24424305 0.76 ADRA1A (0.49) ADRA1ANAMPTADRA1DADRA1BKDM4E
SCHEMBL9342154 0.73 KDM4E (0.46) ADRA1AADRA1DADRA1BKDM4ECYP2C19
SCHEMBL30915761 0.73 KDM4E (0.46) ADRA1AADRA1DADRA1BKDM4ECYP2C19
SCHEMBL31133117 0.73 NOTUM (0.37) KDM4ECYP2C19NOTUMNEK2GABRP
SCHEMBL17338866 0.73 PDPK1 (0.41) KDM4ECYP2C19NOTUMCDK9GABRP
SCHEMBL23641525 0.73 ADRA1A (0.40) ADRA1ANAMPTADRA1DADRA1BCDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114929697-A Azabenzimidazole compounds and medicaments 日本新药株式会社 2022-08-19 CN claimed
CN-114929697-A Azabenzimidazole compounds and medicaments 日本新药株式会社 2022-08-19 CN disclosed
US-5547961-A USING TETRAHYDROIMIDAZOPYRIDINE YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1996-08-20 US disclosed
US-5336679-A Treatment of irritable bowel syndrome YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1994-08-09 US disclosed
EP-0532754-A1 TETRAHYDROIMIDAZOPYRIDINE DERIVATIVE OR ITS SALT YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1993-03-24 EP disclosed