SCHEMBL8987490

SCHEMBL8987490

O=C(O)CCCN(Cc1cccc(Cl)c1)Cc1cccc(Cl)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.53
TSHR P16473 2/20 0.50
RECQL P46063 1/20 0.50
KMT2A Q03164 3/20 0.49
ALDH1A1 P00352 2/20 0.49
HDAC3 O15379 2/20 0.46
HDAC1 Q13547 2/20 0.46
HDAC2 Q92769 2/20 0.46
HDAC8 Q9BY41 2/20 0.46
NCOR2 Q9Y618 2/20 0.46
FFAR4 Q5NUL3 1/20 0.45
MEN1 O00255 1/20 0.45
HTT P42858 1/20 0.45
THRA P10827 1/20 0.45
THRB P10828 1/20 0.45
RIPK1 Q13546 1/20 0.45
CTBP2 P56545 1/20 0.44
TAS2R14 Q9NYV8 1/20 0.44
PLAAT3 P53816 1/20 0.43
PLAAT5 Q96KN8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8425195 0.83 TSHR (0.51) TSHRRECQLKMT2AALDH1A1HTT
SCHEMBL1830778 0.82 HDAC3 (0.63) SMN1; SMN2HDAC3HDAC1HDAC2HDAC8
SCHEMBL8987604 0.82 KMT2A (0.64) SMN1; SMN2KMT2AHDAC3HDAC1HDAC2
SCHEMBL8987696 0.81 HDAC3 (0.46) SMN1; SMN2TSHRALDH1A1HDAC3HDAC1
Hydrochloric Acid SCHEMBL8987622 0.80 HDAC3 (0.61) SMN1; SMN2HDAC3HDAC1HDAC2HDAC8
SCHEMBL8987493 0.80 FFAR1 (0.47) SMN1; SMN2TSHRKMT2AALDH1A1HDAC3
SCHEMBL5024832 0.79 SMN1; SMN2 (0.68) SMN1; SMN2KMT2AALDH1A1HDAC3HDAC1
SCHEMBL6508483 0.79 TSHR (0.45) SMN1; SMN2TSHRRECQLKMT2AALDH1A1
SCHEMBL15862571 0.79 HDAC3 (0.58) SMN1; SMN2HDAC3HDAC1HDAC2HDAC8
SCHEMBL7829175 0.78 SMN1; SMN2 (0.67) SMN1; SMN2KMT2AALDH1A1HDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0345068-B1 Agonist of gamma-aminobutyric acid WYETH JOHN & BROTHER LTD (GB) 1995-03-15 EP claimed
US-5321047-A Antidepressant JOHN WYETH & BROTHER, LIMITED (GB) 1994-06-14 US claimed
EP-0345068-A2 Agonist of gamma-aminobutyric acid JOHN WYETH & BROTHER LIMITED (GB) 1989-12-06 EP claimed
US-5527955-A AGONIST OF GAMMA AMINOBUTYRIC ACID JOHN WYETH & BROTHER, LIMITED (GB) 1996-06-18 US disclosed
EP-0345068-B1 Agonist of gamma-aminobutyric acid WYETH JOHN & BROTHER LTD (GB) 1995-03-15 EP disclosed
EP-0345068-A2 Agonist of gamma-aminobutyric acid JOHN WYETH & BROTHER LIMITED (GB) 1989-12-06 EP disclosed