SCHEMBL8990439

SCHEMBL8990439

NC(=O)c1ccc2[nH]cc(C3=CCC(NCCc4ccccc4)CC3)c2c1

nearest known ligand 0.82

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 10/20 0.82
HTR1E P28566 2/20 0.78
HTR1A P08908 1/20 0.78
NOS3 P29474 4/20 0.47
NOS1 P29475 4/20 0.47
SLC6A2 P23975 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9166018 0.95 HTR1D (0.83) HTR1DHTR1EHTR1ANOS3NOS1
SCHEMBL9164512 0.91 HTR1D (0.79) HTR1DHTR1EHTR1ANOS3NOS1
SCHEMBL8990483 0.91 HTR1D (0.67) HTR1DHTR1EHTR1ANOS3NOS1
SCHEMBL9166468 0.91 HTR1D (0.79) HTR1DHTR1EHTR1ANOS3NOS1
SCHEMBL9228535 0.90 HTR1D (0.74) HTR1DHTR1EHTR1ANOS3NOS1
SCHEMBL9253801 0.89 HTR1D (0.65) HTR1DHTR1EHTR1ANOS3NOS1
SCHEMBL9228014 0.89 HTR1D (0.65) HTR1DHTR1EHTR1ANOS3NOS1
SCHEMBL9163972 0.89 HTR1D (0.75) HTR1DHTR1EHTR1ANOS3NOS1
SCHEMBL9160928 0.89 HTR1D (0.64) HTR1DHTR1EHTR1ANOS3NOS1
SCHEMBL9166041 0.88 HTR1D (0.64) HTR1DHTR1EHTR1ANOS3NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5468768-A FOR TREATING VASCULAR HEADACHES BRISTOL-MYERS SQUIBB COMPANY (US) 1995-11-21 US claimed
EP-0666258-A1 Indolylcycloaklanylamin- und Indolylcycloalkenylamine derivatives, their preparation and their use as anti-migraine agents Bristol-Myers Squibb Company (US) 1995-08-09 EP claimed
US-5583149-A TREATING VASCULAR HEADACHES BRISTOL-MYERS SQUIBB COMPANY (US) 1996-12-10 US disclosed
US-5468768-A FOR TREATING VASCULAR HEADACHES BRISTOL-MYERS SQUIBB COMPANY (US) 1995-11-21 US disclosed
EP-0666258-A1 Indolylcycloaklanylamin- und Indolylcycloalkenylamine derivatives, their preparation and their use as anti-migraine agents Bristol-Myers Squibb Company (US) 1995-08-09 EP disclosed