SCHEMBL9228014

SCHEMBL9228014

COC(=O)c1ccc2[nH]cc(C3=CCC(NCCc4ccccc4)CC3)c2c1

nearest known ligand 0.67

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 10/20 0.65
HTR1E P28566 2/20 0.62
HTR1A P08908 1/20 0.62
SLC6A2 P23975 2/20 0.44
NOS3 P29474 2/20 0.44
NOS1 P29475 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8990483 0.91 HTR1D (0.67) HTR1DHTR1EHTR1ASLC6A2NOS3
SCHEMBL9253801 0.90 HTR1D (0.65) HTR1DHTR1EHTR1ASLC6A2NOS3
SCHEMBL8990439 0.89 HTR1D (0.82) HTR1DHTR1EHTR1ASLC6A2NOS3
SCHEMBL9163214 0.88 HTR1D (0.63) HTR1DHTR1EHTR1ASLC6A2NOS3
SCHEMBL9160928 0.87 HTR1D (0.64) HTR1DHTR1EHTR1ASLC6A2NOS3
SCHEMBL8990411 0.85 HTR1D (0.60) HTR1DHTR1EHTR1ASLC6A2NOS3
SCHEMBL9166018 0.84 HTR1D (0.83) HTR1DHTR1EHTR1ASLC6A2NOS3
SCHEMBL9163972 0.84 HTR1D (0.75) HTR1DHTR1EHTR1ASLC6A2NOS3
SCHEMBL8990392 0.83 HTR1D (0.57) HTR1DHTR1EHTR1ASLC6A2NOS3
SCHEMBL9166041 0.83 HTR1D (0.64) HTR1DHTR1EHTR1ASLC6A2NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0666258-A1 Indolylcycloaklanylamin- und Indolylcycloalkenylamine derivatives, their preparation and their use as anti-migraine agents Bristol-Myers Squibb Company (US) 1995-08-09 EP disclosed