SCHEMBL8990601

SCHEMBL8990601

CCCCCc1ccc(-c2ccc(CCc3ccc(C(F)(F)F)cc3)cc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.56
RARB P10826 6/20 0.51
HSD17B10 Q99714 2/20 0.51
TSHR P16473 1/20 0.51
FDFT1 P37268 2/20 0.51
ALDH1A1 P00352 2/20 0.50
RARA P10276 2/20 0.50
MEN1 O00255 1/20 0.50
MAPT P10636 1/20 0.50
MTOR P42345 1/20 0.50
KMT2A Q03164 1/20 0.50
FAAH O00519 1/20 0.49
TAAR1 Q96RJ0 1/20 0.48
HRH3 Q9Y5N1 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
ESR1 P03372 2/20 0.47
ADRA2A P08913 2/20 0.47
ADORA3 P0DMS8 2/20 0.47
TACR2 P21452 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17108417 0.98 MAOB (0.58) MAOBRARBHSD17B10TSHRFDFT1
SCHEMBL10382748 0.98 MAOB (0.58) MAOBRARBHSD17B10TSHRFDFT1
SCHEMBL10382373 0.96 MAOB (0.56) MAOBRARBHSD17B10TSHRFDFT1
SCHEMBL10381424 0.96 MAOB (0.56) MAOBRARBHSD17B10TSHRFDFT1
SCHEMBL10382743 0.96 MAOB (0.56) MAOBRARBHSD17B10TSHRFDFT1
SCHEMBL10381425 0.96 MAOB (0.56) MAOBRARBHSD17B10TSHRFDFT1
SCHEMBL10381412 0.96 MAOB (0.56) MAOBRARBHSD17B10TSHRFDFT1
SCHEMBL10382742 0.96 MAOB (0.56) MAOBRARBHSD17B10TSHRFDFT1
SCHEMBL8990675 0.95 MAOB (0.58) MAOBRARBHSD17B10TSHRFDFT1
SCHEMBL9352104 0.94 TAAR1 (0.53) MAOBHSD17B10ALDH1A1FAAHTAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5496499-A Biphenylethanes and liquid-crystalline phase MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-03-05 US disclosed
EP-0429558-B1 DIPHENYLYLETHANES AND LIQUID CRYSTALLINE PHASE MERCK PATENT GMBH (DE) 1994-03-30 EP disclosed
WO-1990008757-A1 DIPHENYLYLETHANES AND LIQUID CRYSTALLINE PHASE MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1990-08-09 WO disclosed