SCHEMBL8990714

SCHEMBL8990714

CCCCc1ccc(CCc2ccc(-c3ccc(Cl)c(F)c3)cc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RARB P10826 10/20 0.54
RARA P10276 2/20 0.54
RARG P13631 1/20 0.54
AKR1C2 P52895 1/20 0.48
AKR1C1 Q04828 1/20 0.48
HRH3 Q9Y5N1 1/20 0.41
CTRC Q99895 1/20 0.41
TSHR P16473 1/20 0.41
HSD17B10 Q99714 1/20 0.41
KCNH2 Q12809 2/20 0.40
MAPT P10636 2/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
MTOR P42345 1/20 0.40
KMT2A Q03164 1/20 0.40
HTR2A P28223 1/20 0.40
FFAR1 O14842 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7764845 0.95 RARB (0.59) RARBRARARARGAKR1C2AKR1C1
SCHEMBL7772878 0.90 RARB (0.46) RARBRARARARGAKR1C2AKR1C1
SCHEMBL30466107 0.88 RARB (0.47) RARBRARARARGAKR1C2AKR1C1
SCHEMBL8857916 0.88 RARB (0.47) RARBRARARARGAKR1C2AKR1C1
SCHEMBL3162001 0.88 RARB (0.46) RARBRARARARGAKR1C2AKR1C1
SCHEMBL7770631 0.87 TAAR1 (0.42) RARBRARARARGKCNH2HTR2A
SCHEMBL8448249 0.86 RARB (0.45) RARBRARARARGAKR1C2AKR1C1
SCHEMBL8448252 0.86 RARB (0.45) RARBRARARARGAKR1C2AKR1C1
SCHEMBL3152588 0.86 RARB (0.44) RARBRARARARGAKR1C2AKR1C1
SCHEMBL9329602 0.85 RARB (0.57) RARBRARARARGAKR1C2AKR1C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5496499-A Biphenylethanes and liquid-crystalline phase MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-03-05 US disclosed
EP-0429558-B1 DIPHENYLYLETHANES AND LIQUID CRYSTALLINE PHASE MERCK PATENT GMBH (DE) 1994-03-30 EP disclosed
WO-1990008757-A1 DIPHENYLYLETHANES AND LIQUID CRYSTALLINE PHASE MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1990-08-09 WO disclosed