SCHEMBL8991749

SCHEMBL8991749

C=Cc1cccc(S(=O)(=O)O)c1C(C)C

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.36
TTR P02766 1/20 0.35
TDP1 Q9NUW8 2/20 0.35
KDM4E B2RXH2 1/20 0.34
MYC P01106 1/20 0.33
SLC9A1 P19634 1/20 0.33
AHR P35869 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7755428 0.78 CYP1A2 (0.35) CYP1A2TTRTDP1MYCSLC9A1
SCHEMBL8335964 0.77 MYC (0.40) CYP1A2TTRTDP1MYCSLC9A1
SCHEMBL8991753 0.77 CYP1A2 (0.35) CYP1A2TTRTDP1SLC9A1
SCHEMBL2543853 0.77 TTR (0.40) CYP1A2TTRTDP1MYCSLC9A1
SCHEMBL438031 0.77 TTR (0.40) CYP1A2TTRTDP1MYCSLC9A1
SCHEMBL8991792 0.76 CYP1A2 (0.37) CYP1A2TTRTDP1MYCSLC9A1
SCHEMBL15000 0.76 TDP1 (0.44) CYP1A2TTRTDP1MYCSLC9A1
SCHEMBL29361804 0.76 TDP1 (0.44) CYP1A2TTRTDP1MYCSLC9A1
SCHEMBL10423504 0.75 AURKA (0.41) CYP1A2TTRTDP1KDM4EMYC
SCHEMBL2553027 0.75 GABRA1 (0.43) CYP1A2TTRMYC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530317-B1 CROSS-LINKED CONDUCTIVE POLYMERS AND ANTISTAT COATINGS EMPLOYING THE SAME EASTMAN KODAK CO (US) 1996-07-31 EP disclosed
EP-0530316-B1 CROSS-LINKED CONDUCTIVE POLYMERS AND ANTISTAT LAYERS EMPLOYING THE SAME EASTMAN KODAK CO (US) 1995-01-25 EP disclosed
US-5318878-A Cross-linked conductive polymers and antistat layers employing the same EASTMAN KODAK COMPANY (US) 1994-06-07 US disclosed
US-5198499-A CROSS-LINKED POLYMERS FROM VINYL BENZENE SULFONATE SALTS, ETHYLENIC HYDROXY MONOMERS AND HYDROXYL CONTAINING BINDER POLYMERS EASTMAN KODAK COMPANY (US) 1993-03-30 US disclosed
EP-0530316-A1 CROSS-LINKED CONDUCTIVE POLYMERS AND ANTISTAT LAYERS EMPLOYING THE SAME. EASTMAN KODAK CO (US) 1993-03-10 EP disclosed
EP-0530317-A1 CROSS-LINKED CONDUCTIVE POLYMERS AND ANTISTAT COATINGS EMPLOYING THE SAME. EASTMAN KODAK CO (US) 1993-03-10 EP disclosed
US-5126405-A Coatings for photographic films EASTMAN KODAK COMPANY (US) 1992-06-30 US disclosed
US-5096975-A CROSS-LINKED POLYMERS FROM VINYL BENZENE SULFONATE SALTS AND ETHYLENIC HYDROXY MONOMERS EASTMAN KODAK COMPANY (US) 1992-03-17 US disclosed
WO-1991018062-A1 CROSS-LINKED CONDUCTIVE POLYMERS AND ANTISTAT COATINGS EMPLOYING THE SAME EASTMAN KODAK COMPANY (US) 1991-11-28 WO disclosed
WO-1991018061-A1 CROSS-LINKED CONDUCTIVE POLYMERS AND ANTISTAT LAYERS EMPLOYING THE SAME EASTMAN KODAK COMPANY (US) 1991-11-28 WO disclosed