SCHEMBL8992521

SCHEMBL8992521

COC(=O)C=C1C=CCN1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.39
KEAP1 Q14145 1/20 0.33
NFE2L2 Q16236 1/20 0.33
HCAR2 Q8TDS4 1/20 0.33
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
CA12 O43570 1/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
TYR P14679 1/20 0.30
CA7 P43166 1/20 0.30
CA9 Q16790 1/20 0.30
CA14 Q9ULX7 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11726683 0.66 TSHR (0.49) TSHRKEAP1NFE2L2HCAR2MEN1
SCHEMBL28857840 0.65 HCAR2 (0.36) TSHRKEAP1NFE2L2HCAR2MEN1
SCHEMBL518574 0.62
SCHEMBL23087147 0.62 HCAR2 (0.46) TSHRKEAP1NFE2L2HCAR2MEN1
SCHEMBL23087148 0.62 HCAR2 (0.46) TSHRKEAP1NFE2L2HCAR2MEN1
SCHEMBL4954055 0.60 TSHR (0.44) TSHRKEAP1NFE2L2HCAR2
SCHEMBL4954046 0.60 TSHR (0.44) TSHRKEAP1NFE2L2HCAR2
SCHEMBL9612293 0.60 TSHR (0.44) TSHRKEAP1NFE2L2HCAR2
SCHEMBL1035256 0.60 TSHR (0.43) TSHRKEAP1NFE2L2HCAR2MEN1
SCHEMBL8190673 0.59 TSHR (0.42) TSHRKEAP1NFE2L2HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5541327-A Preparation of camptothecin analogs SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1996-07-30 US disclosed
US-5525731-A CYCLIZATION; HALOGENATION; ALKYLATION; REDUCTION; HYDROLYSIS; DECARBOXYLATION; SELENYLATION SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1996-06-11 US disclosed
US-5446047-A Anticancer agents SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1995-08-29 US disclosed
US-5391745-A Cytotoxic activity towards cancer cells SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1995-02-21 US disclosed