SCHEMBL8992901

SCHEMBL8992901

Cc1cc(C(C)(C)C)cc(CO[SiH](C)C)c1Br

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 3/20 0.34
CYP1A2 P05177 2/20 0.34
CYP2D6 P10635 2/20 0.34
CYP2C9 P11712 2/20 0.34
HIF1A Q16665 1/20 0.34
HTR1D P28221 2/20 0.33
POLB P06746 1/20 0.33
GABRA1 P14867 1/20 0.31
GABRB2 P47870 1/20 0.31
HTR1B P28222 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8536110 0.77 CYP2D6 (0.36) CYP2C19CYP1A2CYP2D6CYP2C9HIF1A
SCHEMBL1086377 0.71 POLB (0.52) CYP2C19CYP1A2CYP2D6CYP2C9HIF1A
SCHEMBL914375 0.71 CYP2C19 (0.40) CYP2C19CYP1A2CYP2D6CYP2C9HIF1A
SCHEMBL7904051 0.70 CYP2D6 (0.36) CYP2C19CYP1A2CYP2D6
SCHEMBL4589689 0.70 CYP2D6 (0.54) CYP2C19CYP1A2CYP2D6HIF1A
SCHEMBL916519 0.69 CYP2D6 (0.39) CYP2C19CYP1A2CYP2D6CYP2C9HIF1A
SCHEMBL914352 0.68 CYP2C19 (0.38) CYP2C19CYP1A2CYP2D6CYP2C9HIF1A
SCHEMBL6940383 0.68 PTGDR2 (0.42)
SCHEMBL914908 0.67 PTPN1 (0.42) CYP2C19CYP1A2CYP2D6CYP2C9HIF1A
SCHEMBL9127939 0.66 CYP2D6 (0.31) CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516777-A PROSTATE CANCER THERAPY OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-05-14 US disclosed
US-5409928-A Prostate diseases, alopecia OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-04-25 US disclosed
EP-0594149-A2 Condensed pyrazole derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-04-27 EP disclosed