SCHEMBL8995518

SCHEMBL8995518

Fc1ccc(-c2ccc(I)s2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 5/20 0.48
HSD17B2 P37059 5/20 0.48
RAB9A P51151 3/20 0.44
KDM4E B2RXH2 2/20 0.44
NPC1 O15118 2/20 0.44
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
MAPT P10636 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
MAPK14 Q16539 1/20 0.40
APP P05067 3/20 0.39
ESR1 P03372 2/20 0.39
ESR2 Q92731 2/20 0.39
ESRRG P62508 3/20 0.39
PTPN2 P17706 1/20 0.39
PTPN11 Q06124 1/20 0.39
FLT3 P36888 1/20 0.38
PRF1 P14222 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12581415 0.83 HSD17B1 (0.63) HSD17B1HSD17B2RAB9AKDM4ENPC1
SCHEMBL12980677 0.81 APP (0.42) HSD17B1HSD17B2RAB9AMEN1KMT2A
SCHEMBL12562851 0.80 HSD17B1 (0.61) HSD17B1HSD17B2RAB9AKDM4ENPC1
SCHEMBL12562796 0.80 HSD17B1 (0.61) HSD17B1HSD17B2RAB9AKDM4ENPC1
SCHEMBL12562798 0.78 HSD17B1 (0.59) HSD17B1HSD17B2RAB9AKDM4ENPC1
SCHEMBL12562792 0.78 HSD17B1 (0.59) HSD17B1HSD17B2RAB9AKDM4ENPC1
SCHEMBL9933404 0.78 HSD17B1 (0.59) HSD17B1HSD17B2RAB9AKDM4ENPC1
SCHEMBL12562788 0.78 HSD17B1 (0.59) HSD17B1HSD17B2RAB9AKDM4ENPC1
SCHEMBL15243106 0.77 APP (0.44) HSD17B1HSD17B2APPESR1ESR2
SCHEMBL4843589 0.77 APP (0.39) HSD17B1HSD17B2RAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016041470-A1 SGLT-2 INHIBITORS NATIONAL INSTITUTE OF BIOLOGICAL SCIENCES, BEIJING (CN) 2016-03-24 WO disclosed
EP-2530079-A1 PHENYL C-GLUCOSIDE DERIVATIVES, PREPARATION METHODS AND USES THEREOF Tianjin Institute Of Pharmaceutical Research (CN) 2012-12-05 EP disclosed
US-5580989-A Process for the preparation of N-4-[(substituted phenyl)alkylheterocyclic]-N ABBOTT LABORATORIES (US) 1996-12-03 US disclosed
EP-0726897-A1 PROCESS FOR THE PREPARATION OF N-4- (SUBSTITUTED PHENYL)ALKYLTHIENYL]-, AND N-4- (SUBSTITUTED PHENYL)ALKYLFURYL]BUT-3-YN-2-YL]-N-HYDROXYUREA COMPOUNDS Abbott Laboratories (US) 1996-08-21 EP disclosed
WO-1995012589-A1 PROCESS FOR THE PREPARATION OF N-4-[(SUBSTITUTED PHENYL)ALKYLTHIENYL]-, AND N-4-[(SUBSTITUTED PHENYL)ALKYLFURYL]BUT-3-YN-2-YL]-N-HYDROXYUREA COMPOUNDS ABBOTT LABORATORIES (US) 1995-05-11 WO disclosed