SCHEMBL8997154

SCHEMBL8997154

CCOC(=O)CC[C@H](NC(=O)c1ccc(C(C)CCC2CNc3nc(N)nc(N)c32)cc1)C(=O)OCC

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DHFR P00374 4/20 0.48
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
HSD17B10 Q99714 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
ATIC P31939 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8997160 1.00 DHFR (0.48) DHFRKDM4EALDH1A1HPGDHSD17B10
SCHEMBL8997237 0.87 DHFR (0.50) DHFRKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9041263 0.87 DHFR (0.50) DHFRKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9041254 0.87 DHFR (0.50) DHFRKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9041638 0.87 DHFR (0.48) DHFRKDM4EALDH1A1HPGDHSD17B10
SCHEMBL8997230 0.87 DHFR (0.50) DHFRKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9040997 0.87 DHFR (0.48) DHFRKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9040986 0.87 DHFR (0.48) DHFRKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9042233 0.86 DHFR (0.54) DHFRKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9042227 0.86 DHFR (0.54) DHFRKDM4EALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4997838-A Antitumor agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1991-03-05 US claimed
EP-0334636-B1 Pyrrolopyrimidine derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1996-10-23 EP disclosed
US-5539113-A ANTITUMOR AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-07-23 US disclosed
US-5296600-A Antitumor agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-03-22 US disclosed
US-5106974-A Antitumor and -carcinogenic agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-04-21 US disclosed
US-4997838-A Antitumor agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1991-03-05 US disclosed
EP-0334636-A2 Pyrrolopyrimidine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1989-09-27 EP disclosed