SCHEMBL8997255

SCHEMBL8997255

Nc1nc(O)c2c(CCCc3ccc(C(=O)N[C@H](CCC(=O)O)C(=O)O)cc3)c[nH]c2n1

nearest known ligand 0.75

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DHFR P00374 9/20 0.75
TYMS P04818 5/20 0.75
GART P22102 7/20 0.66
FOLR1 P15328 5/20 0.66
SLC46A1 Q96NT5 5/20 0.66
SLC19A1 P41440 4/20 0.66
FOLR2 P14207 3/20 0.66
ATIC P31939 2/20 0.66
SHMT1 P34896 1/20 0.66
FRK P42685 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8997171 1.00 DHFR (0.75) DHFRTYMSGARTFOLR1SLC46A1
SCHEMBL9223619 0.97 DHFR (0.70) DHFRTYMSGARTFOLR1SLC46A1
Pemetrexed SCHEMBL7848273 0.95 DHFR (0.83) DHFRTYMSGARTFOLR1SLC46A1
Pemetrexed SCHEMBL12022769 0.95 DHFR (0.83) DHFRTYMSGARTFOLR1SLC46A1
SCHEMBL5300564 0.92 DHFR (0.76) DHFRTYMSGARTFOLR1SLC46A1
SCHEMBL7835435 0.92 DHFR (0.76) DHFRTYMSGARTFOLR1SLC46A1
SCHEMBL9227343 0.91 DHFR (0.78) DHFRTYMSGARTFOLR1SLC46A1
SCHEMBL9227108 0.91 DHFR (0.78) DHFRTYMSGARTFOLR1SLC46A1
SCHEMBL9085671 0.91 DHFR (0.75) DHFRTYMSGARTFOLR1SLC46A1
SCHEMBL8997183 0.90 DHFR (0.76) DHFRTYMSGARTFOLR1SLC46A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5539113-A ANTITUMOR AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-07-23 US disclosed
US-5496946-A Production of pyrrolopyrimidines and intermediates therefor TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-03-05 US disclosed
US-5349064-A Production of pyrrolopyrimidines TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-09-20 US disclosed
EP-0402903-A1 Production of pyrrolopyrimidines and intermediates therefor Takeda Chemical Industries, Ltd. (JP) 1990-12-19 EP disclosed