SCHEMBL8997538

SCHEMBL8997538

COC(=O)C=C(C)NC1CC1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.38
HCAR2 Q8TDS4 2/20 0.37
KEAP1 Q14145 1/20 0.37
NFE2L2 Q16236 1/20 0.37
POLB P06746 2/20 0.36
NPSR1 Q6W5P4 1/20 0.36
TSHR P16473 2/20 0.36
EPHX2 P34913 3/20 0.35
MMP2 P08253 1/20 0.34
MMP8 P22894 1/20 0.34
EPHX1 P07099 5/20 0.34
MAPT P10636 2/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8984934 1.00 SMN1; SMN2 (0.38) SMN1; SMN2HCAR2KEAP1NFE2L2POLB
SCHEMBL10560406 0.92 NPSR1 (0.46) SMN1; SMN2POLBNPSR1EPHX2EPHX1
SCHEMBL10560424 0.92 NPSR1 (0.46) SMN1; SMN2POLBNPSR1EPHX2EPHX1
SCHEMBL4381636 0.90 NPSR1 (0.49) SMN1; SMN2POLBNPSR1EPHX2EPHX1
SCHEMBL4381639 0.90 NPSR1 (0.49) SMN1; SMN2POLBNPSR1EPHX2EPHX1
SCHEMBL2082055 0.81 NPSR1 (0.44) HCAR2NPSR1TSHREPHX1MAPT
SCHEMBL2082056 0.81 NPSR1 (0.44) HCAR2NPSR1TSHREPHX1MAPT
SCHEMBL1242806 0.74 LMNA (0.43) NPSR1TSHRMMP2EPHX1MAPT
SCHEMBL1242807 0.74 LMNA (0.43) NPSR1TSHRMMP2EPHX1MAPT
SCHEMBL10561685 0.73 LMNA (0.45) NPSR1MMP2EPHX1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-6179654-A None JP disclosed
US-5559139-A ANTIISCHEMIC AGENTS, MICROCIRCULATION BAYER AKTIENGESELLSCHAFT (DE) 1996-09-24 US disclosed
JP-H06179654-A 1,4-DIHYDROPYRIDINE-3,5-DICARBOXYLIC ACID ESTER BAYER AG 1994-06-28 JP disclosed