SCHEMBL8998961

SCHEMBL8998961

O=C(O)C(Cc1c[nH]c2ccccc12)NC(=O)C(F)(F)F

nearest known ligand 0.74

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ACE P12821 4/20 0.74
ALOX15 P16050 1/20 0.67
ITGB2 P05107 5/20 0.66
ICAM1 P05362 5/20 0.66
ITGAL P20701 5/20 0.66
ECE1 P42892 3/20 0.60
FPR2 P25090 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11379169 1.00 ACE (0.74) ACEALOX15ITGB2ICAM1ITGAL
SCHEMBL5189433 0.88 ACE (0.82) ACEALOX15ITGB2ICAM1ITGAL
SCHEMBL8466953 0.88 ACE (0.82) ACEALOX15ITGB2ICAM1ITGAL
SCHEMBL28621122 0.87 KMT2A (0.66) ACE
SCHEMBL22216055 0.86 ACE (0.80) ACEALOX15ITGB2ICAM1ITGAL
SCHEMBL8999413 0.86 EGFR (0.64) ACE
SCHEMBL8999055 0.86 EGFR (0.64) ACE
SCHEMBL3857226 0.85 ALOX15 (0.74) ACEALOX15ITGB2ICAM1ITGAL
SCHEMBL3857229 0.85 ALOX15 (0.74) ACEALOX15ITGB2ICAM1ITGAL
SCHEMBL31606494 0.85 ACE (0.79) ACEALOX15ITGB2ICAM1ITGAL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4283337-A Process for the purification of tryptophane and derivatives of tryptophane DEUTSCHE GOLD UND- SILBER-SCHEIDEANSTALT VORMALS ROESSLER (DE) 1981-08-11 US claimed
US-5556874-A ENZYME INHIBITORS AS ANTICARCINOGENIC AGENTS WARNER LAMBERT COMPANY (US) 1996-09-17 US disclosed
US-5464861-A Anticarcinogenic agents WARNER-LAMBERT (US) 1995-11-07 US disclosed
EP-0654024-A1 2-THIOINDOLES (SELENOINDOLES) AND RELATED DISULFIDES (SELENIDES) WHICH INHIBIT PROTEIN TYROSINE KINASES AND WHICH HAVE ANTITUMOR PROPERTIES WARNER-LAMBERT COMPANY (US) 1995-05-24 EP disclosed
WO-1994003427-A1 2-THIOINDOLES (SELENOINDOLES) AND RELATED DISULFIDES (SELENIDES) WHICH INHIBIT PROTEIN TYROSINE KINASES AND WHICH HAVE ANTITUMOR PROPERTIES WARNER-LAMBERT COMPANY (US) 1994-02-17 WO disclosed
US-4283337-A Process for the purification of tryptophane and derivatives of tryptophane DEUTSCHE GOLD UND- SILBER-SCHEIDEANSTALT VORMALS ROESSLER (DE) 1981-08-11 US disclosed