SCHEMBL9001827

SCHEMBL9001827

CCC(CCn1ccc2nc(N)[nH]c(=O)c21)c1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)s1

nearest known ligand 0.71

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ATIC P31939 14/20 0.71
SHMT1 P34896 14/20 0.71
SHMT2 P34897 14/20 0.71
GART P22102 13/20 0.70
FOLR1 P15328 3/20 0.49
DHFR P00374 1/20 0.49
TYMS P04818 1/20 0.49
SLC19A1 P41440 1/20 0.48
SLC46A1 Q96NT5 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9001782 0.93 ATIC (0.68) ATICSHMT1SHMT2GARTFOLR1
SCHEMBL9001790 0.91 ATIC (0.73) ATICSHMT1SHMT2GARTFOLR1
SCHEMBL9001823 0.88 ATIC (0.55) ATICSHMT1SHMT2GARTFOLR1
SCHEMBL9001763 0.86 ATIC (0.69) ATICSHMT1SHMT2GARTFOLR1
SCHEMBL8571212 0.86 ATIC (0.53) ATICSHMT1SHMT2GARTDHFR
SCHEMBL8571222 0.86 ATIC (0.53) ATICSHMT1SHMT2GARTDHFR
SCHEMBL9001755 0.86 ATIC (0.73) ATICSHMT1SHMT2GARTDHFR
SCHEMBL9001824 0.85 ATIC (0.91) ATICSHMT1SHMT2GARTFOLR1
SCHEMBL9001757 0.84 ATIC (0.66) ATICSHMT1SHMT2GARTFOLR1
SCHEMBL9001783 0.84 ATIC (0.75) ATICSHMT1SHMT2GARTFOLR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed
EP-0530579-A1 Condensed pyrimidine derivatives antitumor agents Eisai Co., Ltd. (JP) 1993-03-10 EP disclosed