SCHEMBL9002014

SCHEMBL9002014

Cc1cn2c(SCCN)cccc2n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2D6 P10635 2/20 0.35
CYP2C9 P11712 2/20 0.35
CYP2C19 P33261 2/20 0.35
STAT6 P42226 1/20 0.35
MAPT P10636 6/20 0.35
SMN1; SMN2 Q16637 6/20 0.35
RAB9A P51151 2/20 0.35
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
NPC1 O15118 1/20 0.35
ALPL P05186 1/20 0.34
TP53 P04637 1/20 0.34
KDM4E B2RXH2 2/20 0.33
HTT P42858 2/20 0.32
MAPK1 P28482 2/20 0.32
ALDH1A1 P00352 3/20 0.32
GAA P10253 2/20 0.32
DDAH1 O94760 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7835501 0.81 SMN1; SMN2 (0.35) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL9002023 0.72 CDK8 (0.42) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL5658100 0.72 CYP3A4 (0.37) CYP3A4MAPTSMN1; SMN2RAB9AKMT2A
Hydrochloric Acid SCHEMBL9001976 0.71 CDK8 (0.41)
SCHEMBL7835026 0.70 KMT2A (0.39) MAPTSMN1; SMN2KMT2ATP53KDM4E
SCHEMBL3448499 0.70 PDE10A (0.41) MAPTSMN1; SMN2RAB9AKMT2AMEN1
SCHEMBL8373773 0.70 ALDH1A1 (0.40) SMN1; SMN2RAB9AKMT2ANPC1KDM4E
SCHEMBL7947747 0.69 GAA (0.50) MAPTSMN1; SMN2RAB9AKMT2AMEN1
Bromide SCHEMBL7844571 0.68 PDE10A (0.40) MAPTSMN1; SMN2RAB9AKMT2AMEN1
SCHEMBL15004601 0.66 RAB9A (0.38) MAPTSMN1; SMN2RAB9AKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5587383-A CALMODULIN INHIBITORS; ANTIISCHEMIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-12-24 US disclosed
EP-0471236-B1 Imidazopyridine derivatives and their use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-03-15 EP disclosed
US-5395839-A Calmodulin and angiogenesis inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-03-07 US disclosed
US-5244908-A Calmodulin inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-09-14 US disclosed
EP-0471236-A1 Imidazopyridine derivatives and their use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-02-19 EP disclosed