SCHEMBL9002335

SCHEMBL9002335

CC(C)OC(=O)N(C)CCSc1cccc2nccn12

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 1/20 0.34
POLB P06746 1/20 0.34
HTT P42858 1/20 0.34
KMT2A Q03164 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
CDK8 P49336 2/20 0.31
ROCK1 Q13464 2/20 0.31
FLT1 P17948 1/20 0.31
CDK9 P50750 1/20 0.31
LIMK1 P53667 1/20 0.31
CLK4 Q9HAZ1 1/20 0.31
CHEK1 O14757 1/20 0.31
MAP4K4 O95819 1/20 0.31
CSF1R P07333 1/20 0.31
PRKACA P17612 1/20 0.31
KDR P35968 1/20 0.31
MAP2K1 Q02750 1/20 0.31
ACVR1 Q04771 1/20 0.31
MAP4K2 Q12851 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9002450 0.87 ALDH1A1 (0.33) ALDH1A1KDM4EPOLBHTTKMT2A
SCHEMBL9002396 0.83 CDK8 (0.34) ALDH1A1KDM4EKMT2ACDK8ROCK1
SCHEMBL9002524 0.80 CDK8 (0.31) ALDH1A1KDM4EPOLBHTTCDK8
SCHEMBL9001960 0.78 CDK8 (0.34) CDK8ROCK1FLT1CDK9LIMK1
Hydrochloric Acid SCHEMBL9001979 0.78 SMN1; SMN2 (0.36) ALDH1A1KDM4EPOLBHTTKMT2A
SCHEMBL9002391 0.78 CDK8 (0.32) CDK8ROCK1FLT1CDK9LIMK1
SCHEMBL9001914 0.77 BRD4 (0.36) ALDH1A1KDM4EPOLBHTTKMT2A
SCHEMBL9002374 0.77 BRD4 (0.38) ALDH1A1KDM4EPOLBHTTKMT2A
SCHEMBL9002463 0.75 CDK8 (0.35) CDK8ROCK1FLT1CDK9LIMK1
Hydrochloric Acid SCHEMBL9185489 0.74 CDK8 (0.34) CDK8ROCK1FLT1CDK9LIMK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5587383-A CALMODULIN INHIBITORS; ANTIISCHEMIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-12-24 US disclosed
EP-0471236-B1 Imidazopyridine derivatives and their use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-03-15 EP disclosed
US-5395839-A Calmodulin and angiogenesis inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-03-07 US disclosed
US-5244908-A Calmodulin inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-09-14 US disclosed
EP-0471236-A1 Imidazopyridine derivatives and their use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-02-19 EP disclosed