SCHEMBL9002425

SCHEMBL9002425

O=S(=O)(NCCCCOc1cccc2nccn12)C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.40
NPY5R Q15761 1/20 0.39
EPHX1 P07099 1/20 0.37
F13A1 P00488 4/20 0.34
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
EGLN1 Q9GZT9 1/20 0.33
CDK8 P49336 2/20 0.33
ROCK1 Q13464 2/20 0.33
CHEK1 O14757 1/20 0.33
MAP4K4 O95819 1/20 0.33
CSF1R P07333 1/20 0.33
PRKACA P17612 1/20 0.33
KDR P35968 1/20 0.33
MAP2K1 Q02750 1/20 0.33
ACVR1 Q04771 1/20 0.33
MAP4K2 Q12851 1/20 0.33
DYRK1A Q13627 1/20 0.33
AURKB Q96GD4 1/20 0.33
DYRK1B Q9Y463 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9002271 0.99 NPY5R (0.41) IDO1NPY5REPHX1F13A1CNR1
SCHEMBL9002354 0.99 NPY5R (0.41) IDO1NPY5REPHX1F13A1CNR1
SCHEMBL9001957 0.96 IDO1 (0.43) IDO1NPY5REPHX1F13A1CNR1
SCHEMBL9001878 0.93 IDO1 (0.39) IDO1NPY5REPHX1EGLN1CDK8
SCHEMBL9002403 0.84 CYP4F2 (0.41) NPY5RF13A1CDK8ROCK1CHEK1
SCHEMBL9001970 0.83 CYP4F2 (0.42) NPY5RF13A1CDK8ROCK1CHEK1
SCHEMBL9002264 0.83 CYP4F2 (0.42) NPY5RF13A1CDK8ROCK1CHEK1
SCHEMBL9001991 0.81 POLB (0.38) NPY5RF13A1CDK8ROCK1CHEK1
SCHEMBL7863546 0.81 NPY5R (0.39) IDO1NPY5REPHX1F13A1CNR1
SCHEMBL7872382 0.80 NPY5R (0.40) IDO1NPY5REPHX1F13A1CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5587383-A CALMODULIN INHIBITORS; ANTIISCHEMIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-12-24 US disclosed
EP-0471236-B1 Imidazopyridine derivatives and their use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-03-15 EP disclosed
US-5395839-A Calmodulin and angiogenesis inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-03-07 US disclosed
US-5244908-A Calmodulin inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-09-14 US disclosed
EP-0471236-A1 Imidazopyridine derivatives and their use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-02-19 EP disclosed