SCHEMBL9001970

SCHEMBL9001970

CS(=O)(=O)NCCCCCOc1cccc2nccn12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 1/20 0.42
CYP4A11 Q02928 1/20 0.42
NPY5R Q15761 4/20 0.38
F13A1 P00488 4/20 0.37
POLB P06746 1/20 0.37
CDK8 P49336 2/20 0.34
ROCK1 Q13464 2/20 0.34
CHEK1 O14757 1/20 0.34
MAP4K4 O95819 1/20 0.34
CSF1R P07333 1/20 0.34
PRKACA P17612 1/20 0.34
KDR P35968 1/20 0.34
MAP2K1 Q02750 1/20 0.34
ACVR1 Q04771 1/20 0.34
MAP4K2 Q12851 1/20 0.34
DYRK1A Q13627 1/20 0.34
AURKB Q96GD4 1/20 0.34
DYRK1B Q9Y463 1/20 0.34
FLT1 P17948 1/20 0.34
CDK9 P50750 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9002264 1.00 CYP4F2 (0.42) CYP4F2CYP4A11NPY5RF13A1POLB
SCHEMBL9002403 0.99 CYP4F2 (0.41) CYP4F2CYP4A11NPY5RF13A1POLB
SCHEMBL9001991 0.95 POLB (0.38) CYP4F2CYP4A11NPY5RF13A1POLB
SCHEMBL9002512 0.91 HTT (0.41) POLBCDK8ROCK1CHEK1MAP4K4
SCHEMBL9002354 0.85 NPY5R (0.41) CYP4F2CYP4A11NPY5RF13A1CDK8
SCHEMBL9002271 0.85 NPY5R (0.41) CYP4F2CYP4A11NPY5RF13A1CDK8
SCHEMBL9002425 0.83 IDO1 (0.40) CYP4F2CYP4A11NPY5RF13A1CDK8
SCHEMBL7841691 0.82 KDM4E (0.41) CDK8ROCK1CHEK1MAP4K4CSF1R
SCHEMBL9002497 0.80 ALDH1A1 (0.54) NPY5RF13A1ALDH1A1TDP1
SCHEMBL9002415 0.80 MAPK1 (0.51) F13A1MEN1HTTKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5587383-A CALMODULIN INHIBITORS; ANTIISCHEMIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-12-24 US disclosed
EP-0471236-B1 Imidazopyridine derivatives and their use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-03-15 EP disclosed
US-5244908-A Calmodulin inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-09-14 US disclosed
EP-0471236-A1 Imidazopyridine derivatives and their use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-02-19 EP disclosed