SCHEMBL9004933

SCHEMBL9004933

C[C@@H]1O[C@@]1(Cn1cncn1)c1ccccc1Cl

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 7/20 0.44
THRB P10828 1/20 0.44
CYP19A1 P11511 2/20 0.41
CYP2C9 P11712 2/20 0.40
GAA P10253 1/20 0.38
HSD17B10 Q99714 1/20 0.38
KDM4E B2RXH2 3/20 0.38
HSP90AA1 P07900 3/20 0.36
NPSR1 Q6W5P4 1/20 0.36
POLB P06746 1/20 0.35
HTT P42858 1/20 0.35
NR1I2 O75469 1/20 0.35
LMNA P02545 1/20 0.35
FYN P06241 1/20 0.35
PGR P06401 1/20 0.35
CHRM2 P08172 1/20 0.35
CHRM4 P08173 1/20 0.35
CHRM5 P08912 1/20 0.35
ADRA2A P08913 1/20 0.35
CHRM1 P11229 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9195837 0.89 CYP3A4 (0.42) CYP3A4THRBCYP19A1CYP2C9GAA
SCHEMBL9195834 0.89 CYP3A4 (0.42) CYP3A4THRBCYP19A1CYP2C9GAA
SCHEMBL8815519 0.85 CYP3A4 (0.61) CYP3A4THRBCYP2C9KDM4EHSP90AA1
SCHEMBL8815515 0.85 CYP3A4 (0.61) CYP3A4THRBCYP2C9KDM4EHSP90AA1
SCHEMBL8781569 0.84 MAPK1 (0.40) CYP3A4THRBCYP19A1CYP2C9GAA
SCHEMBL7655138 0.84 MAPK1 (0.40) CYP3A4THRBCYP19A1CYP2C9GAA
SCHEMBL20621487 0.81 GAA (0.50) CYP3A4THRBCYP19A1GAAHSD17B10
SCHEMBL3467654 0.80 CYP3A4 (0.48) CYP3A4THRBCYP19A1CYP2C9GAA
SCHEMBL2557411 0.80 CYP3A4 (0.48) CYP3A4THRBCYP19A1CYP2C9GAA
SCHEMBL8813224 0.80 CYP3A4 (0.46) CYP3A4THRBCYP19A1CYP2C9GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5495024-A FUNGICIDES TAKEDA CHEMICAL INDUSTRIES LTD. (JP) 1996-02-27 US disclosed
US-5371100-A An 1-(1H-1,2,4-triazolyl) or 1-(1H-imidazolyl)-2-phenyl-3-(1H or 2H-tetrazolyl)-2-alkylol or alkyloxyacetyl fungicides for fungal infections TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-12-06 US disclosed
EP-0548553-A1 Optically active azole compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1993-06-30 EP disclosed