SCHEMBL9007018

SCHEMBL9007018

C[Si](C)(C)C#CSc1ccc2c(c1)OCCC2

nearest known ligand 0.36

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 8/20 0.36
CTNNB1 P35222 1/20 0.33
WNT3A P56704 1/20 0.33
NOTUM Q6P988 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8566959 0.89 NOTUM (0.41) CTNNB1WNT3ANOTUM
SCHEMBL9486327 0.80 KCNH2 (0.34) KCNH2CTNNB1WNT3ANOTUM
SCHEMBL22098111 0.77 HTR2C (0.39) KCNH2CTNNB1WNT3ANOTUM
SCHEMBL9006824 0.75 CTNNB1 (0.38) KCNH2CTNNB1WNT3A
SCHEMBL5440454 0.73 KCNH2 (0.37) KCNH2CTNNB1WNT3ANOTUM
SCHEMBL6594574 0.72 MAOB (0.39)
SCHEMBL22681792 0.69 HTR2C (0.39) KCNH2CTNNB1WNT3A
SCHEMBL8560705 0.68 DYRK1A (0.41) CTNNB1WNT3ANOTUM
SCHEMBL436669 0.68 KCNH2 (0.49) KCNH2CTNNB1WNT3A
SCHEMBL22681788 0.68 HTR2C (0.43) KCNH2CTNNB1WNT3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0571546-B1 CHROMAN AND THIOCHROMANS WITH PHENYLETHYNYL SUBSTITUENTS AT THE 7-POSITION HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY ALLERGAN INC (US) 1996-10-16 EP disclosed
US-5346915-A Chromans and thiochromans with phenylethynyl substituents at the 7-position having retinold-like biological activity ALLERGAN, INC. (US) 1994-09-13 US disclosed
US-5346895-A Treating dermatoses, immunological disorders, wound healing ALLERGAN, INC. (US) 1994-09-13 US disclosed
EP-0571546-A1 CHROMAN AND THIOCHROMANS WITH PHENYLETHYNYL SUBSTITUENTS AT THE 7-POSITION HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY. ALLERGAN INC (US) 1993-12-01 EP disclosed
WO-1992014725-A1 CHROMAN AND THIOCHROMANS WITH PHENYLETHYNYL SUBSTITUENTS AT THE 7-POSITION HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY ALLERGAN, INC. (US) 1992-09-03 WO disclosed