SCHEMBL9008669

SCHEMBL9008669

NC(=O)N(c1ccc2c(c1)CCC2)[C@H]1N=C(C2CCCCC2)c2ccccc2N(CCN2CCOCC2)C1=O

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 6/20 0.40
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39
KDM4E B2RXH2 1/20 0.37
MAPT P10636 1/20 0.37
CCKBR P32239 6/20 0.36
CCKAR P32238 2/20 0.36
HPGD P15428 1/20 0.36
ALOX15 P16050 1/20 0.36
HTT P42858 1/20 0.36
OXTR P30559 1/20 0.34
CSF1R P07333 1/20 0.34
USP2 O75604 1/20 0.34
CYP3A4 P08684 1/20 0.34
THRB P10828 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9008683 0.87 CCKBR (0.45) BDKRB1CCKBRCCKAR
SCHEMBL9008792 0.87 CCKBR (0.45) BDKRB1CCKBRCCKAR
SCHEMBL9008684 0.81 BDKRB1 (0.45) BDKRB1CCKBRCCKAROXTR
SCHEMBL7592838 0.81 BDKRB1 (0.55) BDKRB1CCKBRCCKAR
SCHEMBL9008659 0.79 CCKBR (0.41) BDKRB1KDM4ECCKBROXTR
SCHEMBL9008744 0.79 CCKBR (0.42) BDKRB1CCKBRCCKAROXTR
SCHEMBL9008853 0.78 BDKRB1 (0.59) BDKRB1CCKBR
SCHEMBL9008785 0.78 EPHX2 (0.41) KDM4ECCKBR
SCHEMBL9008842 0.76 MAPT (0.43) BDKRB1KDM4EMAPTCCKBRCCKAR
SCHEMBL9008676 0.76 MAPT (0.43) BDKRB1KDM4EMAPTCCKBRCCKAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5556969-A Benzodiazepine derivatives MERCK SHARP & DOHME LTD. (GB) 1996-09-17 US claimed