SCHEMBL9010792

SCHEMBL9010792

C#CC(C)(C)NC(=O)c1cccs1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.55
HDAC1 Q13547 1/20 0.55
MEN1 O00255 3/20 0.51
KMT2A Q03164 3/20 0.51
ALOX15 P16050 2/20 0.51
HTT P42858 1/20 0.51
ALDH1A1 P00352 5/20 0.51
RAB9A P51151 9/20 0.50
NPC1 O15118 8/20 0.50
TDP1 Q9NUW8 1/20 0.50
SMN1; SMN2 Q16637 2/20 0.47
KDM4E B2RXH2 1/20 0.47
LMNA P02545 1/20 0.47
HPGD P15428 1/20 0.47
MAPK1 P28482 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
HSD17B10 Q99714 1/20 0.47
MAPT P10636 3/20 0.46
PKM P14618 1/20 0.46
CES2 O00748 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29528205 0.85 CTSC (0.56) TSHRHDAC1MEN1KMT2AALOX15
SCHEMBL4043837 0.82 MEN1 (0.68) TSHRHDAC1MEN1KMT2AALOX15
SCHEMBL15709252 0.81 TSHR (0.50) TSHRHDAC1MEN1KMT2AALOX15
SCHEMBL12497851 0.81 TSHR (0.50) TSHRHDAC1MEN1KMT2AALOX15
SCHEMBL4909498 0.78 GAA (0.47) MEN1KMT2AHTTALDH1A1RAB9A
SCHEMBL30433221 0.77 TSHR (0.59) TSHRHDAC1MEN1KMT2AALOX15
SCHEMBL3229709 0.75 TSHR (0.58) TSHRHDAC1MEN1KMT2AALOX15
SCHEMBL3240216 0.75 TSHR (0.58) TSHRHDAC1MEN1KMT2AALOX15
SCHEMBL3127881 0.75 HDAC1 (0.62) TSHRHDAC1MEN1KMT2AHTT
SCHEMBL4095096 0.74 KDM4E (0.45) TSHRMEN1KMT2AALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5547984-A FUNGICIDES ROHM AND HAAS COMPANY (US) 1996-08-20 US disclosed
US-5529978-A FUNGICIDE ROHM AND HAAS COMPANY (US) 1996-06-25 US disclosed
US-5344978-A Fungicides ROHM AND HAAS COMPANY (US) 1994-09-06 US disclosed
US-5196046-A N-acetonyl-substituted-amides ROHM AND HAAS COMPANY (US) 1993-03-23 US disclosed
EP-0170498-B1 N-ACETONYL-SUBSTITUTED-AMIDES, COMPOSITIONS CONTAINING THEM AND THEIR USE IN COMBATING FUNGI ROHM AND HAAS COMPANY (US) 1991-09-11 EP disclosed
US-4863940-A N-acetonyl-substituted amides and phytopathogenic fungicidal use thereof ROHM AND HAAS (US) 1989-09-05 US disclosed
EP-0170498-A2 N-acetonyl-substituted-amides, compositions containing them and their use in combating fungi ROHM AND HAAS COMPANY (US) 1986-02-05 EP disclosed