SCHEMBL9011282

SCHEMBL9011282

CN1C=C(C(=O)NCCCC(=O)OCc2ccccc2)Cc2ccccc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.45
HTT P42858 1/20 0.44
HSP90AA1 P07900 2/20 0.43
EPHX2 P34913 1/20 0.43
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
TPSAB1 Q15661 2/20 0.40
TPSD1 Q9BZJ3 2/20 0.40
TPSG1 Q9NRR2 2/20 0.40
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
NAMPT P43490 1/20 0.40
KEAP1 Q14145 1/20 0.39
NFE2L2 Q16236 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8509550 0.78 HTT (0.44) HTTHSP90AA1EPHX2MEN1KMT2A
SCHEMBL12409527 0.71 HTT (0.80) HTTEPHX2MEN1KMT2ATPSAB1
SCHEMBL24180428 0.70 HTT (0.60) HTTHSP90AA1EPHX2MEN1KMT2A
SCHEMBL13251782 0.70 HTT (0.64) HTTHSP90AA1EPHX2MEN1KMT2A
SCHEMBL17787475 0.70 LTA4H (0.56) HTTHSP90AA1EPHX2MEN1KMT2A
SCHEMBL4767870 0.70 NOTUM (0.44) NOTUMMEN1KMT2ACYP3A4ALDH1A1
SCHEMBL19996577 0.69 ATM (0.68) HTTEPHX2MEN1KMT2ACYP3A4
Hydrochloric Acid SCHEMBL25244621 0.69 LTA4H (0.54) HTTHSP90AA1EPHX2MEN1KMT2A
SCHEMBL13991918 0.69 HTT (0.55) HTTHSP90AA1EPHX2MEN1KMT2A
SCHEMBL2898427 0.69 HTT (0.56) HTTEPHX2MEN1KMT2ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5525727-A ANALGESIC OR NARCOTIC ANTAGONIST UNIVERSITY OF FLORIDA (US) 1996-06-11 US disclosed
US-5187158-A Sustained delivery of viricides UNIVERSITY OF FLORIDA (US) 1993-02-16 US disclosed
US-5008257-A Penicillin or cephalosporin antibiotics UNIVERSITY OF FLORIDA (US) 1991-04-16 US disclosed
US-4900837-A Brain-specific drug delivery of steroid sex hormones cleaved from pyridinium carboxylates and dihydro-pyridine carboxylate precursors UNIVERSITY OF FLORIDA (US) 1990-02-13 US disclosed
US-4880921-A Brain-specific drug delivery UNIVERSITY OF FLORIDA (US) 1989-11-14 US disclosed
US-4824850-A DIHYDROPYRIDINE-PYRIDINIUM SALT REDOX CARRIER UNIVERSITY OF FLORIDA (US) 1989-04-25 US disclosed