Iodide

Iodide

SCHEMBL9011297

C[n+]1cccc(C(=O)NCCc2ccc(OC(=O)C(C)(C)C)c(OC(=O)C(C)(C)C)c2)c1.[I-]

nearest known ligand 0.44

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHRM1CHRM3CHRNA1CHRNB1CHRNDCHRNECHRNG

The experimentally established mechanism targets of Iodide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.44
GAA P10253 2/20 0.43
ALDH1A1 P00352 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
HPGD P15428 1/20 0.42
ALOX12 P18054 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
CA14 Q9ULX7 1/20 0.42
ESRRG P62508 1/20 0.42
MAPT P10636 2/20 0.41
APOBEC3A P31941 2/20 0.40
APOBEC3G Q9HC16 2/20 0.40
KDM4E B2RXH2 1/20 0.40
POLB P06746 1/20 0.40
PABPC1 P11940 1/20 0.40
LMNA P02545 1/20 0.39
MEN1 O00255 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL9011417 0.93 CA1 (0.41) MAPK1GAAALDH1A1SMN1; SMN2HPGD
Iodide SCHEMBL9011351 0.89 TRPV1 (0.50) MAPK1GAAALDH1A1SMN1; SMN2HPGD
Iodide SCHEMBL9011303 0.86 SMN1; SMN2 (0.47) GAAALDH1A1SMN1; SMN2ESRRGMAPT
Trifluoroacetic Acid SCHEMBL8724650 0.80 ADRB2 (0.50) MAPK1GAAALDH1A1SMN1; SMN2HPGD
Iodide SCHEMBL9011306 0.80 CA1 (0.52) MAPK1GAAALDH1A1SMN1; SMN2HPGD
SCHEMBL9011252 0.79 MAPK1 (0.71) MAPK1GAAALDH1A1SMN1; SMN2MAPT
Iodide SCHEMBL8722463 0.78 MEN1 (0.56) MAPK1GAAALDH1A1HPGDCA1
SCHEMBL9011198 0.77 MEN1 (0.57) MAPK1GAAALDH1A1HPGDCA1
Iodide SCHEMBL9011248 0.77 ESRRG (0.54) GAASMN1; SMN2ESRRGMAPTAPOBEC3A
SCHEMBL21510386 0.76 ADRB2 (0.49) ALDH1A1SMN1; SMN2CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5525727-A ANALGESIC OR NARCOTIC ANTAGONIST UNIVERSITY OF FLORIDA (US) 1996-06-11 US disclosed
US-5187158-A Sustained delivery of viricides UNIVERSITY OF FLORIDA (US) 1993-02-16 US disclosed
US-4900837-A Brain-specific drug delivery of steroid sex hormones cleaved from pyridinium carboxylates and dihydro-pyridine carboxylate precursors UNIVERSITY OF FLORIDA (US) 1990-02-13 US disclosed
US-4880816-A Brain-specific delivery of dopamine utilizing dihydropyridine/pyridinium salt-type redox carriers UNIVERSITY OF FLORIDA (US) 1989-11-14 US disclosed
US-4880921-A Brain-specific drug delivery UNIVERSITY OF FLORIDA (US) 1989-11-14 US disclosed
US-4824850-A DIHYDROPYRIDINE-PYRIDINIUM SALT REDOX CARRIER UNIVERSITY OF FLORIDA (US) 1989-04-25 US disclosed
US-4727079-A Brain-specific dopaminergic activity involving dihydropyridine carboxamides, dihydroquinoline and isoquinoline carboxamides UNIVERSITY OF FLORIDA (US) 1988-02-23 US disclosed
US-4540564-A DIHYDROPYRIDINE AND/OR PYRIDINIUM SALT REDOX CARRIER UNIVERSITY OF FLORIDA (US) 1985-09-10 US disclosed
US-4479932-A DIHYDROPYRIDINE PYRIDINIUM SALT REDOX CARRIER UNIVERSITY OF FLORIDA (US) 1984-10-30 US disclosed
EP-0110955-A1 BRAIN-SPECIFIC DRUG DELIVERY. UNIV FLORIDA (US) 1984-06-20 EP disclosed
WO-1983003968-A1 BRAIN-SPECIFIC DRUG DELIVERY UNIVERSITY OF FLORIDA (US) 1983-11-24 WO disclosed