SCHEMBL9012815

SCHEMBL9012815

N[C@@H](Cc1ccc(N(CCCl)CCCl)cc1)C(=O)N1CCN(CCC(O)(P(=O)(O)O)P(=O)(O)O)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.49
ALDH1A1 P00352 2/20 0.49
ALOX15 P16050 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
HIF1A Q16665 2/20 0.49
LMNA P02545 2/20 0.49
KMT2A Q03164 2/20 0.49
ABCB11 O95342 1/20 0.49
CHRM2 P08172 1/20 0.49
ADRA2A P08913 1/20 0.49
CHRM1 P11229 1/20 0.49
ACHE P22303 1/20 0.49
PTGS1 P23219 1/20 0.49
OPRM1 P35372 1/20 0.49
DRD3 P35462 1/20 0.49
SLC6A3 Q01959 1/20 0.49
KCNH2 Q12809 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
CYP1A2 P05177 1/20 0.49
NFKB1 P19838 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9012805 0.99 CYP3A4 (0.48) CYP3A4ALDH1A1ALOX15SMN1; SMN2HIF1A
SCHEMBL9012789 0.94 CYP3A4 (0.47) CYP3A4ALDH1A1ALOX15SMN1; SMN2HIF1A
Hydrochloric Acid SCHEMBL9012915 0.94 CYP3A4 (0.47) CYP3A4ALDH1A1ALOX15SMN1; SMN2HIF1A
SCHEMBL9012814 0.89 CYP3A4 (0.42) CYP3A4ALDH1A1ALOX15SMN1; SMN2HIF1A
SCHEMBL9013067 0.88 CYP3A4 (0.42) CYP3A4ALDH1A1ALOX15SMN1; SMN2HIF1A
SCHEMBL9013081 0.88 LMNA (0.44) CYP3A4ALDH1A1ALOX15SMN1; SMN2HIF1A
SCHEMBL9012902 0.86 CYP3A4 (0.48) CYP3A4ALDH1A1ALOX15SMN1; SMN2HIF1A
Hydrochloric Acid SCHEMBL9120139 0.85 CYP3A4 (0.47) CYP3A4ALDH1A1ALOX15SMN1; SMN2HIF1A
SCHEMBL9012823 0.84 CYP3A4 (0.41) CYP3A4ALDH1A1ALOX15SMN1; SMN2HIF1A
SCHEMBL9122764 0.83 CYP3A4 (0.41) CYP3A4ALDH1A1ALOX15SMN1; SMN2HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0580642-B1 AMINOACYL DERIVATIVES OF GEM-DIPHOSPHONIC ACIDS, A PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BOEHRINGER MANNHEIM ITALIA (IT) 1996-11-06 EP disclosed
US-5446187-A Aminoacyl derivatives of gem-diphosphonic acids, a process for the preparation thereof and pharmaceutical compositions containing them BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1995-08-29 US disclosed
WO-1992018512-A1 AMINOACYL DERIVATIVES OF GEM-DIPHOSPHONIC ACIDS, A PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1992-10-29 WO disclosed