SCHEMBL9013121

SCHEMBL9013121

N[C@@H](Cc1ccc(N(CCCl)CCCl)cc1)C(=O)N[C@@H](CCC(=O)NCCCC(O)(P(=O)(O)O)P(=O)(O)O)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.47
ALDH1A1 P00352 3/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
HIF1A Q16665 3/20 0.47
LMNA P02545 3/20 0.47
ALOX15 P16050 2/20 0.47
KMT2A Q03164 2/20 0.47
NFKB1 P19838 2/20 0.47
THPO P40225 2/20 0.47
MAPT P10636 2/20 0.47
PMP22 Q01453 2/20 0.47
ABCB11 O95342 1/20 0.47
CHRM2 P08172 1/20 0.47
ADRA2A P08913 1/20 0.47
CHRM1 P11229 1/20 0.47
ACHE P22303 1/20 0.47
PTGS1 P23219 1/20 0.47
OPRM1 P35372 1/20 0.47
DRD3 P35462 1/20 0.47
SLC6A3 Q01959 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9012816 0.98 CYP3A4 (0.46) CYP3A4ALDH1A1SMN1; SMN2HIF1ALMNA
SCHEMBL9013070 0.86 CA12 (0.49) ALDH1A1SMN1; SMN2HIF1ALMNAKMT2A
SCHEMBL8983269 0.85 CYP3A4 (0.53) CYP3A4ALDH1A1SMN1; SMN2HIF1ALMNA
SCHEMBL9012853 0.85 CYP3A4 (0.48) CYP3A4ALDH1A1SMN1; SMN2HIF1ALMNA
Hydrochloric Acid SCHEMBL8983345 0.84 CYP3A4 (0.52) CYP3A4ALDH1A1SMN1; SMN2HIF1ALMNA
SCHEMBL9013048 0.84 CYP3A4 (0.47) CYP3A4ALDH1A1SMN1; SMN2HIF1ALMNA
SCHEMBL9012734 0.84 CYP3A4 (0.47) CYP3A4ALDH1A1SMN1; SMN2HIF1ALMNA
SCHEMBL9012862 0.84 CA12 (0.48) ALDH1A1SMN1; SMN2HIF1ALMNAKMT2A
SCHEMBL9012828 0.83 OPRM1 (0.47) CYP3A4ALDH1A1SMN1; SMN2HIF1ALMNA
SCHEMBL9012827 0.83 OPRM1 (0.43) CYP3A4ALDH1A1SMN1; SMN2HIF1ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0580642-B1 AMINOACYL DERIVATIVES OF GEM-DIPHOSPHONIC ACIDS, A PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BOEHRINGER MANNHEIM ITALIA (IT) 1996-11-06 EP disclosed
US-5446187-A Aminoacyl derivatives of gem-diphosphonic acids, a process for the preparation thereof and pharmaceutical compositions containing them BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1995-08-29 US disclosed