SCHEMBL9014740

SCHEMBL9014740

CCOC(=O)COc1cnc2c(n1)CCCC2

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.58
ALDH1A1 P00352 2/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
HSD17B10 Q99714 3/20 0.41
GAA P10253 2/20 0.41
TSHR P16473 2/20 0.40
NLRP3 Q96P20 2/20 0.40
CXCR1 P25024 1/20 0.40
CXCR2 P25025 1/20 0.40
HPGD P15428 1/20 0.40
PARP1 P09874 1/20 0.40
NPSR1 Q6W5P4 1/20 0.39
POLB P06746 1/20 0.39
GLA P06280 1/20 0.38
CA12 O43570 1/20 0.38
CA9 Q16790 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4137212 0.76 KDM4E (0.48) KDM4EALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL2848228 0.72 KDM4E (0.56) KDM4EALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL30075963 0.70 KDM4E (0.50) KDM4EALDH1A1SMN1; SMN2KMT2AHSD17B10
SCHEMBL19555374 0.70 KDM4E (0.50) KDM4EALDH1A1SMN1; SMN2KMT2AHSD17B10
SCHEMBL9014694 0.69 LOX (0.35)
SCHEMBL16837304 0.69 KDM4E (0.56) KDM4EALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL9014882 0.69 KDM4E (0.33) KDM4EALDH1A1TSHR
SCHEMBL9014730 0.68 CYP1A2 (0.32)
SCHEMBL1686063 0.68 ALDH1A1 (0.48) KDM4EALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL19555296 0.68 KDM4E (0.51) KDM4EALDH1A1SMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5578596-A TREATMENT OF SEROTONERGIC NEURON RELATED DISEASES, MOTION SICKNESS, ANXIXETY, DEPRESSION ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1996-11-26 US disclosed
EP-0668276-A1 2-ALKOXY-5,6,7,8-TETRAHYDROQUINOXALINE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1995-08-23 EP disclosed