SCHEMBL9017041

SCHEMBL9017041

COc1ccc(Nc2ncnc3cc(C(F)(F)F)ccc23)cc1

nearest known ligand 0.63

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EGFR P00533 12/20 0.63
LCK P06239 2/20 0.63
MAPT P10636 1/20 0.62
GRM1 Q13255 1/20 0.62
NPC1 O15118 1/20 0.61
HTT P42858 1/20 0.61
RAB9A P51151 1/20 0.61
SMN1; SMN2 Q16637 1/20 0.61
GAK O14976 1/20 0.61
NCOA1 Q15788 1/20 0.58
NCOA3 Q9Y6Q9 1/20 0.58
ABCG2 Q9UNQ0 2/20 0.58
KDR P35968 3/20 0.56
CSF1R P07333 1/20 0.56
TRPV1 Q8NER1 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11094065 0.99 EGFR (0.64) EGFRLCKMAPTGRM1NPC1
SCHEMBL5740105 0.88 EGFR (0.69) EGFRHTTRAB9AGAKABCG2
SCHEMBL11088081 0.83 EGFR (0.69) EGFRLCKHTTABCG2KDR
Hydrochloric Acid SCHEMBL11085999 0.82 TSHR (0.70) EGFRLCKHTTABCG2KDR
SCHEMBL5864703 0.81 EGFR (0.84) EGFRLCKGAKABCG2KDR
Hydrochloric Acid SCHEMBL8808833 0.81 EGFR (0.68) EGFRMAPTNPC1HTTRAB9A
SCHEMBL11083409 0.81 EGFR (0.67) EGFRLCKMAPTGRM1NPC1
SCHEMBL22137768 0.81 TTBK1 (0.61) EGFRGAKKDRCSF1RTRPV1
Hydrochloric Acid SCHEMBL11086239 0.80 EGFR (0.68) EGFRLCKMAPTGRM1NPC1
Hydrochloric Acid SCHEMBL10496016 0.78 EGFR (0.54) EGFRHTTGAKABCG2KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0520722-B1 Therapeutic preparations containing quinazoline derivatives ZENECA LTD (GB) 1996-12-27 EP claimed
EP-0520722-B1 Therapeutic preparations containing quinazoline derivatives ZENECA LTD (GB) 1996-12-27 EP disclosed
US-4464375-A ANALGESIC, ANTIINFLAMMATORY SANKYO CO., LTD. (JP) 1984-08-07 US disclosed
US-4322420-A Method of using 4-anilinoquinazoline derivatives as analgesic and anti-inflammatory agents SANKYO COMPANY LIMITED (JP) 1982-03-30 US disclosed