SCHEMBL9020827

SCHEMBL9020827

C[N+]1(CC2=C(C(=O)O)N3C(=O)C(NC=O)C3SC2)CCN(c2c(F)cc3c(=O)c(C(=O)O)cn(CCF)c3c2F)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 0.54
ALDH1A1 P00352 6/20 0.40
HPGD P15428 6/20 0.40
HSD17B10 Q99714 6/20 0.40
PMP22 Q01453 1/20 0.40
ADRA2B P18089 1/20 0.37
MAPK1 P28482 1/20 0.37
ALB P02768 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
POLB P06746 2/20 0.35
TUBB4A P04350 1/20 0.35
TUBB P07437 1/20 0.35
TUBA3C P0DPH7 1/20 0.35
TUBA1B P68363 1/20 0.35
TUBA4A P68366 1/20 0.35
TUBB4B P68371 1/20 0.35
TUBB3 Q13509 1/20 0.35
TUBB2A Q13885 1/20 0.35
TUBB8 Q3ZCM7 1/20 0.35
TUBA3E Q6PEY2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL9396259 0.96 KDM4E (0.49) KDM4EALDH1A1HPGDHSD17B10PMP22
Trifluoroacetic Acid SCHEMBL9396266 0.96 KDM4E (0.49) KDM4EALDH1A1HPGDHSD17B10PMP22
Iodide SCHEMBL9396283 0.92 KDM4E (0.48) KDM4EALDH1A1HPGDHSD17B10PMP22
Iodide SCHEMBL9022564 0.92 KDM4E (0.48) KDM4EALDH1A1HPGDHSD17B10PMP22
Iodide SCHEMBL9397810 0.86 KDM4E (0.48) KDM4EALDH1A1HPGDHSD17B10PMP22
Iodide SCHEMBL9020946 0.86 KDM4E (0.48) KDM4EALDH1A1HPGDHSD17B10PMP22
Water SCHEMBL9397892 0.86 KDM4E (0.48) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL9744140 0.84 KDM4E (0.56) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL9744130 0.84 KDM4E (0.56) KDM4EALDH1A1HPGDHSD17B10PMP22
Trifluoroacetic Acid SCHEMBL9395038 0.79 NR1I2 (0.32) KDM4EALDH1A1HPGDHSD17B10ADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0335297-B1 Cephalosporin derivatives HOFFMANN LA ROCHE (CH) 1996-03-13 EP claimed