SCHEMBL9022397

SCHEMBL9022397

CCOC(=O)CCCN1CC[C@H](NC(=O)c2cc(Cl)c(N)cc2OC)[C@@H](OC)C1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 15/20 0.74
KCNH2 Q12809 8/20 0.74
CYP3A4 P08684 3/20 0.69
CYP2D6 P10635 3/20 0.69
CYP2C9 P11712 2/20 0.69
USP2 O75604 1/20 0.69
HTR3E A5X5Y0 1/20 0.69
MLNR O43193 1/20 0.69
CACNA1F O60840 1/20 0.69
HTR3B O95264 1/20 0.69
HMGCR P04035 1/20 0.69
HTR1A P08908 1/20 0.69
ADRA2A P08913 1/20 0.69
DRD2 P14416 1/20 0.69
ADRA2B P18089 1/20 0.69
ADRA2C P18825 1/20 0.69
DRD1 P21728 1/20 0.69
TBXA2R P21731 1/20 0.69
ADRA1D P25100 1/20 0.69
HTR2A P28223 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9021703 1.00 HTR4 (0.74) HTR4KCNH2CYP3A4CYP2D6CYP2C9
SCHEMBL9021715 1.00 HTR4 (0.74) HTR4KCNH2CYP3A4CYP2D6CYP2C9
SCHEMBL9022409 1.00 HTR4 (0.74) HTR4KCNH2CYP3A4CYP2D6CYP2C9
SCHEMBL1906067 1.00 HTR4 (0.74) HTR4KCNH2CYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL9022483 0.99 HTR4 (0.73) HTR4KCNH2CYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL9022487 0.99 HTR4 (0.73) HTR4KCNH2CYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL9022491 0.99 HTR4 (0.73) HTR4KCNH2CYP3A4CYP2D6CYP2C9
SCHEMBL735940 0.97 HTR4 (0.72) HTR4KCNH2CYP3A4CYP2D6CYP2C9
SCHEMBL30094488 0.97 HTR4 (0.72) HTR4KCNH2CYP3A4CYP2D6CYP2C9
SCHEMBL13566537 0.97 HTR4 (0.72) HTR4KCNH2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640601-B1 BENZAMIDE DERIVATIVE HOKURIKU PHARMACEUTICAL (JP) 1996-12-04 EP disclosed
US-5500422-A FOR TREATING GASTROINTESTINAL DISEASES HOKURIKU SEIYAKU CO. LTD. (JP) 1996-03-19 US disclosed
US-5395832-A Gastrointestinal disorders HOKURIKU SEIYAKU CO., LTD. (JP) 1995-03-07 US disclosed
EP-0640601-A1 BENZAMIDE DERIVATIVE HOKURIKU SEIYAKU CO., LTD. (JP) 1995-03-01 EP disclosed