SCHEMBL9023015

SCHEMBL9023015

O=C(O)c1cn(-c2cccc(F)c2F)c2c(F)c(F)c(F)cc2c1=O

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.58
KDM4E B2RXH2 1/20 0.58
POLB P06746 1/20 0.58
HSP90AA1 P07900 1/20 0.58
RXFP1 Q9HBX9 1/20 0.58
TOP1 P11387 3/20 0.53
STAT3 P40763 3/20 0.45
HTT P42858 1/20 0.44
TOP2A P11388 9/20 0.44
TOP2B Q02880 8/20 0.44
HPGD P15428 1/20 0.44
HSD17B10 Q99714 1/20 0.44
CHRM1 P11229 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
RORC P51449 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9047182 0.90 ALDH1A1 (0.64) ALDH1A1KDM4EPOLBHSP90AA1RXFP1
SCHEMBL6214789 0.83 KDM4E (0.65) ALDH1A1KDM4EPOLBHSP90AA1RXFP1
SCHEMBL31435135 0.82 ALDH1A1 (0.64) ALDH1A1KDM4EPOLBHSP90AA1RXFP1
SCHEMBL6220162 0.82 ALDH1A1 (0.64) ALDH1A1KDM4EPOLBHSP90AA1RXFP1
SCHEMBL9869652 0.81 ALDH1A1 (0.63) ALDH1A1KDM4EPOLBHSP90AA1RXFP1
SCHEMBL10635691 0.81 ALDH1A1 (0.63) ALDH1A1KDM4EPOLBHSP90AA1RXFP1
SCHEMBL6213800 0.80 ALDH1A1 (0.67) ALDH1A1KDM4EPOLBHSP90AA1RXFP1
SCHEMBL7009143 0.79 TOP1 (0.57) ALDH1A1KDM4EPOLBHSP90AA1RXFP1
SCHEMBL9869480 0.79 ALDH1A1 (0.72) ALDH1A1KDM4EPOLBHSP90AA1RXFP1
SCHEMBL10372132 0.79 ALDH1A1 (0.65) ALDH1A1KDM4EPOLBHSP90AA1RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0500835-B1 A NOVEL QUINOLONE CARBOXYLIC ACID DERIVATIVE DAE WOONG PHARMA (KR) 1996-12-27 EP disclosed