SCHEMBL9024508

SCHEMBL9024508

CC(C)(N)CC(=O)NC1CSc2ccccc2N(Cc2ccc(-c3ccccc3C(N)=O)cc2)C1=O

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 4/20 0.53
AGTR1 P30556 1/20 0.53
XIAP P98170 1/20 0.47
F7 P08709 7/20 0.44
F3 P13726 7/20 0.44
F2 P00734 3/20 0.44
MME P08473 3/20 0.41
ACE P12821 3/20 0.41
PPARG P37231 1/20 0.39
F10 P00742 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9024510 1.00 GHSR (0.53) GHSRAGTR1XIAPF7F3
SCHEMBL7796021 0.87 GHSR (0.53) GHSRAGTR1XIAPF7F3
SCHEMBL9105221 0.87 GHSR (0.42) GHSRAGTR1XIAPF7F3
SCHEMBL9105226 0.87 GHSR (0.42) GHSRAGTR1XIAPF7F3
SCHEMBL7785847 0.85 GHSR (0.51) GHSRAGTR1XIAPF7F3
SCHEMBL9222685 0.85 GHSR (0.51) GHSRAGTR1XIAPF7F3
SCHEMBL7785912 0.85 GHSR (0.51) GHSRAGTR1XIAPF7F3
SCHEMBL9087316 0.85 GHSR (0.58) GHSRAGTR1XIAPF7F3
SCHEMBL9089411 0.85 GHSR (0.56) GHSRAGTR1XIAPF7F3
SCHEMBL9024310 0.85 GHSR (0.72) GHSRAGTR1XIAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0513974-B1 Novel benzo-fused lactams that promote the release of growth hormone MERCK & CO INC (US) 1996-09-04 EP claimed
EP-0513974-A1 Novel benzo-fused lactams that promote the release of growth hormone MERCK & CO. INC. (US) 1992-11-19 EP claimed
US-5310737-A Benzo-fused lactams that promote the release of growth hormone MERCK & CO., INC. (US) 1994-05-10 US disclosed
US-5206235-A Animal growth regulators; stimulants MERCK & CO., INC. (US) 1993-04-27 US disclosed