SCHEMBL9024865

SCHEMBL9024865

CCCCc1nc(-c2cccnc2)cn1Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9277132 0.92
SCHEMBL9113229 0.91 AGTR1 (0.49)
SCHEMBL9024040 0.90 AGTR1 (0.49)
SCHEMBL9238862 0.89
SCHEMBL9116560 0.87 AGTR1 (0.51)
SCHEMBL9115514 0.86
SCHEMBL9024994 0.86
SCHEMBL9025079 0.85
SCHEMBL9024518 0.85
SCHEMBL9024761 0.84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5587390-A Imidazole derivatives having a II antagonist activity ISTITUTO LUSO FARMACO D'ITALIA S.P.A. (IT) 1996-12-24 US claimed
EP-0654030-B1 IMIDAZOLE DERIVATIVES HAVING ANGIOTENSIN II ANTAGONIST ACTIVITY LUSO FARMACO INST (IT) 1996-12-18 EP claimed
EP-0654030-A1 IMIDAZOLE DERIVATIVES HAVING A II ANTAGONIST ACTIVITY. LUSO FARMACO INST (IT) 1995-05-24 EP claimed
WO-1994003449-A1 IMIDAZOLE DERIVATIVES HAVING A II ANTAGONIST ACTIVITY ISTITUTO LUSO FARMACO D'ITALIA S.P.A. (IT) 1994-02-17 WO claimed
US-5587390-A Imidazole derivatives having a II antagonist activity ISTITUTO LUSO FARMACO D'ITALIA S.P.A. (IT) 1996-12-24 US disclosed
EP-0654030-B1 IMIDAZOLE DERIVATIVES HAVING ANGIOTENSIN II ANTAGONIST ACTIVITY LUSO FARMACO INST (IT) 1996-12-18 EP disclosed
WO-1994003449-A1 IMIDAZOLE DERIVATIVES HAVING A II ANTAGONIST ACTIVITY ISTITUTO LUSO FARMACO D'ITALIA S.P.A. (IT) 1994-02-17 WO disclosed