SCHEMBL9025533

SCHEMBL9025533

CCNC(=O)c1ccccc1-c1ccc(CN2C(=O)C(NC(=O)CC(C)(C)N)CCc3ccccc32)cc1

nearest known ligand 0.68

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 4/20 0.68
AGTR1 P30556 1/20 0.68
XIAP P98170 10/20 0.51
NPY1R P25929 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9025540 1.00 GHSR (0.68) GHSRAGTR1XIAPNPY1R
SCHEMBL9025700 0.93 GHSR (0.67) GHSRAGTR1XIAPNPY1R
SCHEMBL9025708 0.93 GHSR (0.67) GHSRAGTR1XIAPNPY1R
SCHEMBL9026268 0.92 GHSR (0.66) GHSRAGTR1XIAPNPY1R
SCHEMBL9026278 0.92 GHSR (0.66) GHSRAGTR1XIAPNPY1R
SCHEMBL9023902 0.92 GHSR (0.70) GHSRAGTR1XIAPNPY1R
SCHEMBL9023922 0.92 GHSR (0.70) GHSRAGTR1XIAPNPY1R
SCHEMBL9025039 0.92 GHSR (0.65) GHSRAGTR1XIAPNPY1R
SCHEMBL9025028 0.92 GHSR (0.65) GHSRAGTR1XIAPNPY1R
SCHEMBL9024310 0.90 GHSR (0.72) GHSRAGTR1XIAPNPY1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0513974-B1 Novel benzo-fused lactams that promote the release of growth hormone MERCK & CO INC (US) 1996-09-04 EP claimed
EP-0513974-B1 Novel benzo-fused lactams that promote the release of growth hormone MERCK & CO INC (US) 1996-09-04 EP disclosed
US-5310737-A Benzo-fused lactams that promote the release of growth hormone MERCK & CO., INC. (US) 1994-05-10 US disclosed
US-5206235-A Animal growth regulators; stimulants MERCK & CO., INC. (US) 1993-04-27 US disclosed
EP-0513974-A1 Novel benzo-fused lactams that promote the release of growth hormone MERCK & CO. INC. (US) 1992-11-19 EP disclosed
WO-1992016524-A1 BENZO-FUSED LACTAMS PROMOTE RELEASE OF GROWTH HORMONE MERCK & CO., INC. (US) 1992-10-01 WO disclosed