SCHEMBL9025569

SCHEMBL9025569

CCOC1(OCC)C(COCc2ccccc2)C(COCc2ccccc2)[C@@H]1F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.38
TAAR1 Q96RJ0 1/20 0.33
LMNA P02545 1/20 0.33
BCHE P06276 2/20 0.32
ACHE P22303 2/20 0.32
CA1 P00915 2/20 0.32
CA2 P00918 2/20 0.32
CA7 P43166 2/20 0.32
CA9 Q16790 2/20 0.32
CTSL P07711 1/20 0.32
CTSB P07858 1/20 0.32
CTSK P43235 1/20 0.32
GAA P10253 1/20 0.31
HTR1A P08908 1/20 0.31
ADRA1D P25100 1/20 0.31
ADRA1A P35348 1/20 0.31
ADRA1B P35368 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9025148 1.00 TSHR (0.38) TSHRTAAR1LMNABCHEACHE
SCHEMBL9025602 1.00 TSHR (0.38) TSHRTAAR1LMNABCHEACHE
SCHEMBL9025142 1.00 TSHR (0.38) TSHRTAAR1LMNABCHEACHE
SCHEMBL9025562 1.00 TSHR (0.38) TSHRTAAR1LMNABCHEACHE
SCHEMBL9026603 0.70 TSHR (0.39) TSHRTAAR1LMNABCHEACHE
SCHEMBL9026613 0.70 TSHR (0.39) TSHRTAAR1LMNABCHEACHE
SCHEMBL9026599 0.70 TSHR (0.39) TSHRTAAR1LMNABCHEACHE
SCHEMBL25347431 0.67 TSHR (0.45) TSHRTAAR1LMNABCHEACHE
SCHEMBL9565493 0.67 MMP1 (0.39) TSHRTAAR1LMNA
SCHEMBL9565490 0.67 MMP1 (0.39) TSHRTAAR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0458363-B1 Fluorinated bis(hydroxymethyl) cyclobutyl purines and pyrimidines SQUIBB & SONS INC (US) 1996-02-07 EP disclosed
WO-1991018969-A1 FLUORINATED BIS(HYDROXYMETHYL)CYCLOBUTYL PURINES AND PYRIMIDINES E.R. SQUIBB & SONS, INC. (US) 1991-12-12 WO disclosed
EP-0458363-A1 Fluorinated bis(hydroxymethyl) cyclobutyl purines and pyrimidines E.R. SQUIBB & SONS, INC. (US) 1991-11-27 EP disclosed