SCHEMBL9025720

SCHEMBL9025720

CC(C)(N)CC(=O)NC1CCCc2ccccc2N(Cc2ccc(-c3ccccc3-c3nnn[nH]3)cc2)C1=O

nearest known ligand 0.70

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 4/20 0.70
AGTR1 P30556 1/20 0.70
XIAP P98170 8/20 0.44
NPY1R P25929 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
L-158432 SCHEMBL9023762 0.96 GHSR (0.76) GHSRAGTR1XIAPNPY1R
L-158432 SCHEMBL7417293 0.96 GHSR (0.76) GHSRAGTR1XIAPNPY1R
L-158432 SCHEMBL9108116 0.94 GHSR (0.74) GHSRAGTR1XIAPNPY1R
L-158432 SCHEMBL9023941 0.92 GHSR (0.71) GHSRAGTR1XIAPNPY1R
SCHEMBL9024343 0.91 GHSR (0.65) GHSRAGTR1XIAP
SCHEMBL9024349 0.90 GHSR (0.68) GHSRAGTR1XIAPNPY1R
SCHEMBL9024158 0.89 GHSR (0.66) GHSRAGTR1XIAPNPY1R
SCHEMBL9024548 0.89 GHSR (0.66) GHSRAGTR1XIAPNPY1R
SCHEMBL9024847 0.88 GHSR (0.66) GHSRAGTR1XIAPNPY1R
SCHEMBL9024557 0.88 GHSR (0.66) GHSRAGTR1XIAPNPY1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0513974-B1 Novel benzo-fused lactams that promote the release of growth hormone MERCK & CO INC (US) 1996-09-04 EP disclosed
US-5310737-A Benzo-fused lactams that promote the release of growth hormone MERCK & CO., INC. (US) 1994-05-10 US disclosed
US-5206235-A Animal growth regulators; stimulants MERCK & CO., INC. (US) 1993-04-27 US disclosed
EP-0513974-A1 Novel benzo-fused lactams that promote the release of growth hormone MERCK & CO. INC. (US) 1992-11-19 EP disclosed
WO-1992016524-A1 BENZO-FUSED LACTAMS PROMOTE RELEASE OF GROWTH HORMONE MERCK & CO., INC. (US) 1992-10-01 WO disclosed